The Impact of Insulin on Low-dose Metronomic Vinorelbine and Mafosfamide in Breast Cancer Cells

Anticancer Res. 2021 Mar;41(3):1243-1250. doi: 10.21873/anticanres.14881.

Abstract

Background/aim: Breast cancer (BC) may be affected by diabetes and anti-diabetic medication, as well as its therapeutic agents. Low-dose metronomic chemotherapy (LDMC) is an available treatment option in BC. We investigated the impact of insulin on low-dose metronomic vinorelbine and mafosfamide in BC cell lines.

Materials and methods: Human BC cell lines T-47D, MCF-7, MDA-MB-231, BT-549 and non-tumorigenic breast cell line MCF-10A were exposed to 0.01 μg/ml and 10 μg/ml insulin in combination with low-dose metronomic vinorelbine or mafosfamide. The cell viability was determined after 24-72 hours using 3-(4,5-dimethylthiazol-2-yl)-2,5-diphenyltetrazolium bromide assay.

Results: Insulin, especially at a concentration of 10 μg/ml, seemed to increase viability of vinorelbine-treated hormone receptor-positive BC cells, whereas low-dose mafosfamide treatment tended to be potentiated by insulin in triple-negative cells.

Conclusion: Our findings suggest that insulin may influence the cytotoxic activity of LDMC depending on insulin concentration, type of cytotoxic drug used and BC cell line.

Keywords: Low-dose metronomic chemotherapy; breast cancer; insulin.

MeSH terms

  • Administration, Metronomic
  • Antineoplastic Agents / administration & dosage*
  • Breast Neoplasms / drug therapy*
  • Breast Neoplasms / pathology
  • Cell Line, Tumor
  • Cell Survival / drug effects
  • Cyclophosphamide / administration & dosage
  • Cyclophosphamide / analogs & derivatives*
  • Female
  • Humans
  • Insulin / pharmacology*
  • Vinorelbine / administration & dosage*

Substances

  • Antineoplastic Agents
  • Insulin
  • mafosfamide
  • Cyclophosphamide
  • Vinorelbine