Kv1.3 voltage-gated potassium channels link cellular respiration to proliferation through a non-conducting mechanism

Cell Death Dis. 2021 Apr 7;12(4):372. doi: 10.1038/s41419-021-03627-6.

Abstract

Cellular energy metabolism is fundamental for all biological functions. Cellular proliferation requires extensive metabolic reprogramming and has a high energy demand. The Kv1.3 voltage-gated potassium channel drives cellular proliferation. Kv1.3 channels localise to mitochondria. Using high-resolution respirometry, we show Kv1.3 channels increase oxidative phosphorylation, independently of redox balance, mitochondrial membrane potential or calcium signalling. Kv1.3-induced respiration increased reactive oxygen species production. Reducing reactive oxygen concentrations inhibited Kv1.3-induced proliferation. Selective Kv1.3 mutation identified that channel-induced respiration required an intact voltage sensor and C-terminal ERK1/2 phosphorylation site, but is channel pore independent. We show Kv1.3 channels regulate respiration through a non-conducting mechanism to generate reactive oxygen species which drive proliferation. This study identifies a Kv1.3-mediated mechanism underlying the metabolic regulation of proliferation, which may provide a therapeutic target for diseases characterised by dysfunctional proliferation and cell growth.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Cell Proliferation / physiology
  • Cell Respiration / physiology
  • Humans
  • Kv1.3 Potassium Channel / metabolism*
  • Membrane Potentials
  • Reactive Oxygen Species / metabolism*
  • Transfection

Substances

  • KCNA3 protein, human
  • Kv1.3 Potassium Channel
  • Reactive Oxygen Species