Fingolimod ameliorates imiquimod-induced psoriasiform dermatitis by sequestrating interleukin-17-producing ?d T cells in secondary lymph nodes

J Dermatol Sci. 2021 May;102(2):116-125. doi: 10.1016/j.jdermsci.2021.04.004. Epub 2021 Apr 15.

Abstract

Background: Psoriasis is a chronic inflammatory skin disease. Interleukin (IL)-17A plays a key role in the pathogenesis of psoriasis. Fingolimod, which is available for the treatment of multiple sclerosis, exerts anti-inflammatory effects by sequestrating inflammatory lymphocytes in secondary lymphoid tissues and the thymus. The effect of fingolimod on psoriasis has not been reported yet.

Objective: Our objectives were to investigate the effect of fingolimod on psoriasis utilizing mice with imiquimod (IMQ)-induced psoriasiform dermatitis, and explore the possibility of fingolimod as a therapeutic agent for psoriasis.

Methods: Psoriasiform dermatitis was induced by imiquimod application on murine shaved back skin for six days. Fingolimod prepared in phosphate-buffered saline (PBS), or PBS alone as a control, was administered intraperitoneally daily from days 0 to 5.

Results: Fingolimod ameliorated IMQ-induced psoriasis dermatitis clinically and histologically. On day 6, the mRNA expression level of IL-17A was lower in the skin of fingolimod-treated mice than in that of PBS-treated mice, whereas it was higher in the inguinal lymph nodes of fingolimod-treated mice than in those of PBS-treated mice. Flow cytometric analyses revealed that fingolimod reduced IL-17A-producing ?d T cells infiltrating into the skin, whereas it increased these cells in the inguinal lymph nodes. Fingolimod inhibited egress of Langerhans cells from the skin to lymph nodes.

Conclusion: Our results demonstrated that fingolimod showed effectiveness for IMQ-induced psoriasiform dermatitis by hindering the emigration of IL-17A-producing ?d T cells from the lymph nodes to the skin, and suggest that fingolimod is a promising candidate for the treatment of psoriasis.

Keywords: Fingolimod; Imiquimod; Lymph node; Psoriasis; Sphingosine 1-phosphate.

MeSH terms

  • Animals
  • Disease Models, Animal
  • Down-Regulation / drug effects
  • Down-Regulation / immunology
  • Drug Evaluation, Preclinical
  • Female
  • Fingolimod Hydrochloride / pharmacology*
  • Fingolimod Hydrochloride / therapeutic use
  • Humans
  • Imiquimod / administration & dosage
  • Imiquimod / immunology
  • Interleukin-17 / metabolism
  • Intraepithelial Lymphocytes / drug effects*
  • Intraepithelial Lymphocytes / immunology
  • Intraepithelial Lymphocytes / metabolism
  • Langerhans Cells / immunology
  • Langerhans Cells / metabolism
  • Lymph Nodes / cytology
  • Lymph Nodes / drug effects*
  • Lymph Nodes / immunology
  • Lymph Nodes / metabolism
  • Mice
  • Psoriasis / drug therapy*
  • Psoriasis / immunology
  • Psoriasis / pathology
  • Skin / cytology
  • Skin / drug effects*
  • Skin / immunology
  • Skin / metabolism
  • Up-Regulation / drug effects
  • Up-Regulation / immunology

Substances

  • Interleukin-17
  • Fingolimod Hydrochloride
  • Imiquimod