Co-Oxidative Transformation of Piperine to Piperonal and 3,4-Methylenedioxycinnamaldehyde by a Lipoxygenase from Pleurotus sapidus

Chembiochem. 2021 Oct 1;22(19):2857-2861. doi: 10.1002/cbic.202100183. Epub 2021 Jun 9.

Abstract

The valuable aroma compound piperonal with its vanilla-like olfactory properties is of high interest for the fragrance and flavor industry. A lipoxygenase (LOXPsa 1) of the basidiomycete Pleurotus sapidus was identified to convert piperine, the abundant pungent principle of black pepper (Piper nigrum), to piperonal and a second volatile product, 3,4-methylenedioxycinnamaldehyde, with a vanilla-like odor through an alkene cleavage. The reaction principle was co-oxidation, as proven by its dependence on the presence of linoleic or α-linolenic acid, common substrates of lipoxygenases. Optimization of the reaction conditions (substrate concentrations, reaction temperature and time) led to a 24-fold and 15-fold increase of the piperonal and 3,4-methylenedioxycinnamaldehyde concentration using the recombinant enzyme. Monokaryotic strains showed different concentrations of and ratios between the two reaction products.

Keywords: biotransformations; cleavage reactions; co-oxidation; lipoxygenase; piperonal.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aldehydes / chemistry
  • Aldehydes / metabolism*
  • Alkaloids / chemistry
  • Alkaloids / metabolism*
  • Benzaldehydes / chemistry
  • Benzaldehydes / metabolism*
  • Benzodioxoles / chemistry
  • Benzodioxoles / metabolism*
  • Lipoxygenase / metabolism*
  • Molecular Structure
  • Oxidation-Reduction
  • Piperidines / chemistry
  • Piperidines / metabolism*
  • Pleurotus / enzymology*
  • Polyunsaturated Alkamides / chemistry
  • Polyunsaturated Alkamides / metabolism*

Substances

  • Aldehydes
  • Alkaloids
  • Benzaldehydes
  • Benzodioxoles
  • Piperidines
  • Polyunsaturated Alkamides
  • Lipoxygenase
  • piperonal
  • piperine

Supplementary concepts

  • Pleurotus sapidus