[Nonsteroidal anti-inflammatory agents. V. Synthesis of 1-aryl-5-(1-pyrryl)-pyrazolyl-4-acetic acids with potential anti-inflammatory action]

Farmaco Sci. 1988 Mar;43(3):251-65.
[Article in Italian]

Abstract

The synthesis of 1-aryl-5-(1-pyrryl)pyrazoles bearing at position 4 an acetic or alpha-propionic chain is described. The new compounds can be structurally related to lonazolac and its analogues with analgesic-antiinflammatory activities. When tested pharmacologically in comparison with tolmetin and indomethacin none of the above derivatives showed any appreciable activity.

Publication types

  • English Abstract
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acetates / chemical synthesis*
  • Animals
  • Anti-Inflammatory Agents, Non-Steroidal / chemical synthesis*
  • Male
  • Mice
  • Pyrazoles / chemical synthesis*
  • Rats
  • Rats, Inbred Strains

Substances

  • Acetates
  • Anti-Inflammatory Agents, Non-Steroidal
  • Pyrazoles