Lateral hypothalamus-projecting noradrenergic locus coeruleus pathway modulates binge-like ethanol drinking in male and female TH-ires-cre mice

Neuropharmacology. 2021 Sep 15:196:108702. doi: 10.1016/j.neuropharm.2021.108702. Epub 2021 Jul 8.

Abstract

A growing body of literature implicates noradrenergic (NE) signaling in the modulation of ethanol consumption. However, relatively few studies have detailed specific brain pathways that mediate NE-associated binge-like ethanol consumption. To begin to fill this gap in the literature, male and female C57BL6/J and TH-ires-cre mice underwent pharmacological and chemogenetic testing, respectively, in combination with "drinking in the dark" procedures to model binge-like consumption of ethanol or sucrose solutions. First, we showed that intraperitoneal administration of the NE reuptake inhibitor, reboxetine, blunted binge-like ethanol intake in C57BL6/J mice. Chemogenetic activation of locus coeruleus (LC) tyrosine hydroxylase (TH)-expressing neurons blunted binge-like ethanol intake regardless of sex. Chemogenetic activation of LC projections to the lateral hypothalamus (LH), a region implicated in ethanol consumption, blunted binge-like ethanol drinking without altering sucrose intake in ethanol-experienced or ethanol-naïve mice. In C57BL/6 J mice, LH-targeted microinfusion of an α1-adrenergic receptor (AR) agonist blunted binge-like ethanol intake across both sexes, while LH infusion of a β-AR agonist blunted binge-like ethanol intake in females exclusively. Finally, in mice with high baseline ethanol intake both an α1- AR agonist and an α-2 AR antagonist blunted binge-like ethanol intake. The present results provide novel evidence that increased NE tone in a circuit arising from the LC and projecting to the LH reduces binge-like ethanol drinking in mice, and may represent a novel approach to treating binge or heavy drinking prior to the development of dependence. This article is part of the special Issue on "Neurocircuitry Modulating Drug and Alcohol Abuse".

Keywords: Binge-like drinking; Chemogenetic; Drinking in the dark; Lateral hypothalamus; Mice; Norepinephrine.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adrenergic Uptake Inhibitors / pharmacology*
  • Adrenergic alpha-1 Receptor Agonists / pharmacology
  • Adrenergic alpha-2 Receptor Agonists / pharmacology
  • Adrenergic beta-Agonists / pharmacology
  • Animals
  • Binge Drinking / metabolism*
  • Binge Drinking / physiopathology
  • Central Nervous System Depressants / administration & dosage*
  • Ethanol / administration & dosage*
  • Female
  • Hypothalamic Area, Lateral / drug effects
  • Hypothalamic Area, Lateral / metabolism*
  • Hypothalamic Area, Lateral / physiopathology
  • Locus Coeruleus / drug effects
  • Locus Coeruleus / metabolism*
  • Locus Coeruleus / physiopathology
  • Male
  • Mice
  • Neural Pathways
  • Norepinephrine / metabolism*
  • Reboxetine / pharmacology*
  • Tyrosine 3-Monooxygenase

Substances

  • Adrenergic Uptake Inhibitors
  • Adrenergic alpha-1 Receptor Agonists
  • Adrenergic alpha-2 Receptor Agonists
  • Adrenergic beta-Agonists
  • Central Nervous System Depressants
  • Ethanol
  • Reboxetine
  • Tyrosine 3-Monooxygenase
  • Norepinephrine