A systematic review on efficacy, safety, and treatment-durability of low-dose rituximab for the treatment of Pemphigus: special focus on COVID-19 pandemic concerns

Immunopharmacol Immunotoxicol. 2021 Oct;43(5):507-518. doi: 10.1080/08923973.2021.1953063. Epub 2021 Jul 21.

Abstract

Background: Rituximab is a FDA-approved monoclonal antibody for adults with moderate to severe potentially life-threatening pemphigus vulgaris. Recent studies have focused on assessments of efficacy and safety of low-dose rituximab (<2 gram in each cycle).

Method: Databases were searched from 2010 to 2020 (last update: 1 June 2020).

Result: Nine studies were entered; including180 cases (92: women, 88: men, age range: 9-83 years). The dosages of each Rituximab cycle varied between ultra-low-dose (≤500 mg for a cycle, either multiple infusions or a single infusion), low-dose (2 × 375 mg/m2 or 2 × 500 mg) and modified-dose (3 × 375 mg/m2 or 3 × 500 mg). The efficacy and safety of Rituximab in the studies are known by the recovery time, relapse time, and side events. According to the studies, 2 × 500 can lead to complete remission in a broad range, from 35 to 82%. These differences might be explained by different end-points and variable cumulative corticosteroid dosage after RTX administration. Although the studies showed that low dose RTX is efficient, there are some controversies regarding the choosing low-dose for severe patients.

Conclusion: Considering the effectiveness of low-dose, intermediate dose, and ultra-low-dose protocols of Rituximab in inducing remission in pemphigus disease and considering factors such as cost of therapy, and the need to induce a minimum of immunosuppression for a minimum duration in the COVID-19 pandemic, suggested to use low-dose Rituximab protocol (2 infusions of 500 mg Rituximab: interval of 2 weeks) to induce the remission in mild-to-moderate pemphigus patients.

Keywords: COVID-19; Pemphigus; autoimmune bullous skin disorder; low-dose; rituximab; systematic review; ultra-low-dose; under-standard dose.

Publication types

  • Systematic Review

MeSH terms

  • Adolescent
  • Adult
  • Aged
  • Aged, 80 and over
  • COVID-19 / diagnosis
  • COVID-19 / immunology*
  • COVID-19 / virology
  • Child
  • Female
  • Humans
  • Immunocompromised Host*
  • Immunologic Factors / administration & dosage*
  • Immunologic Factors / adverse effects
  • Male
  • Middle Aged
  • Pemphigus / diagnosis
  • Pemphigus / drug therapy*
  • Pemphigus / immunology
  • Remission Induction
  • Risk Factors
  • Rituximab / administration & dosage*
  • Rituximab / adverse effects
  • SARS-CoV-2 / immunology
  • Treatment Outcome
  • Young Adult

Substances

  • Immunologic Factors
  • Rituximab