Radiation-Induced Phosphorylation of a Prion-Like Domain Regulates Transformation by FUS-CHOP

Cancer Res. 2021 Oct 1;81(19):4939-4948. doi: 10.1158/0008-5472.CAN-20-1497. Epub 2021 Aug 12.

Abstract

Chromosomal translocations generate oncogenic fusion proteins in approximately one-third of sarcomas, but how these proteins promote tumorigenesis is not well understood. Interestingly, some translocation-driven cancers exhibit dramatic clinical responses to therapy, such as radiotherapy, although the precise mechanism has not been elucidated. Here we reveal a molecular mechanism by which the fusion oncoprotein FUS-CHOP promotes tumor maintenance that also explains the remarkable sensitivity of myxoid liposarcomas to radiation therapy. FUS-CHOP interacted with chromatin remodeling complexes to regulate sarcoma cell proliferation. One of these chromatin remodelers, SNF2H, colocalized with FUS-CHOP genome-wide at active enhancers. Following ionizing radiation, DNA damage response kinases phosphorylated the prion-like domain of FUS-CHOP to impede these protein-protein interactions, which are required for transformation. Therefore, the DNA damage response after irradiation disrupted oncogenic targeting of chromatin remodelers required for FUS-CHOP-driven sarcomagenesis. This mechanism of disruption links phosphorylation of the prion-like domain of an oncogenic fusion protein to DNA damage after ionizing radiation and reveals that a dependence on oncogenic chromatin remodeling underlies sensitivity to radiation therapy in myxoid liposarcoma. SIGNIFICANCE: Prion-like domains, which are frequently translocated in cancers as oncogenic fusion proteins that drive global epigenetic changes, confer sensitivity to radiation via disruption of oncogenic interactions.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Binding Sites
  • Cell Line, Tumor
  • Cell Transformation, Neoplastic / genetics*
  • Cell Transformation, Neoplastic / metabolism*
  • Cell Transformation, Neoplastic / radiation effects
  • Chromatin Assembly and Disassembly
  • Chromatin Immunoprecipitation Sequencing
  • Gene Expression Regulation, Neoplastic
  • Humans
  • Oncogene Proteins, Fusion / chemistry
  • Oncogene Proteins, Fusion / genetics*
  • Oncogene Proteins, Fusion / metabolism*
  • Phosphorylation / radiation effects
  • Protein Binding
  • Protein Interaction Domains and Motifs*
  • RNA-Binding Protein FUS / chemistry
  • RNA-Binding Protein FUS / genetics*
  • RNA-Binding Protein FUS / metabolism*
  • Radiation, Ionizing*
  • Sarcoma / etiology
  • Sarcoma / metabolism
  • Sarcoma / pathology
  • Transcription Factor CHOP / chemistry
  • Transcription Factor CHOP / genetics*
  • Transcription Factor CHOP / metabolism*
  • Translocation, Genetic

Substances

  • Oncogene Proteins, Fusion
  • RNA-Binding Protein FUS
  • TLS-CHOP fusion protein, human
  • Transcription Factor CHOP