Large-Scale Screening for Monogenic and Clinically Defined Familial Hypercholesterolemia in Iceland

Arterioscler Thromb Vasc Biol. 2021 Oct;41(10):2616-2628. doi: 10.1161/ATVBAHA.120.315904. Epub 2021 Aug 19.

Abstract

Objective: Familial hypercholesterolemia (FH) is traditionally defined as a monogenic disease characterized by severely elevated LDL-C (low-density lipoprotein cholesterol) levels. In practice, FH is commonly a clinical diagnosis without confirmation of a causative mutation. In this study, we sought to characterize and compare monogenic and clinically defined FH in a large sample of Icelanders. Approach and Results: We whole-genome sequenced 49 962 Icelanders and imputed the identified variants into an overall sample of 166 281 chip-genotyped Icelanders. We identified 20 FH mutations in LDLR, APOB, and PCSK9 with combined prevalence of 1 in 836. Monogenic FH was associated with severely elevated LDL-C levels and increased risk of premature coronary disease, aortic valve stenosis, and high burden of coronary atherosclerosis. We used a modified version of the Dutch Lipid Clinic Network criteria to screen for the clinical FH phenotype among living adult participants (N=79 058). Clinical FH was found in 2.2% of participants, of whom only 5.2% had monogenic FH. Mutation-negative clinical FH has a strong polygenic basis. Both individuals with monogenic FH and individuals with mutation-negative clinical FH were markedly undertreated with cholesterol-lowering medications and only a minority attained an LDL-C target of <2.6 mmol/L (<100 mg/dL; 11.0% and 24.9%, respectively) or <1.8 mmol/L (<70 mg/dL; 0.0% and 5.2%, respectively), as recommended for primary prevention by European Society of Cardiology/European Atherosclerosis Society cholesterol guidelines. Conclusions: Clinically defined FH is a relatively common phenotype that is explained by monogenic FH in only a minority of cases. Both monogenic and clinical FH confer high cardiovascular risk but are markedly undertreated.

Keywords: genetic screening; genetics; hypercholesterolemia; lipids; mutation.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Aged
  • Aged, 80 and over
  • Apolipoprotein B-100 / genetics*
  • Biomarkers / blood
  • Cardiovascular Diseases / diagnosis
  • Cardiovascular Diseases / ethnology
  • Cardiovascular Diseases / genetics*
  • Cardiovascular Diseases / therapy
  • Female
  • Genetic Association Studies
  • Genetic Predisposition to Disease
  • Humans
  • Hydroxymethylglutaryl-CoA Reductase Inhibitors / therapeutic use
  • Hyperlipoproteinemia Type II / diagnosis
  • Hyperlipoproteinemia Type II / drug therapy
  • Hyperlipoproteinemia Type II / ethnology
  • Hyperlipoproteinemia Type II / genetics*
  • Iceland / epidemiology
  • Lipids / blood*
  • Male
  • Middle Aged
  • Mutation*
  • Phenotype
  • Prevalence
  • Prognosis
  • Proprotein Convertase 9 / genetics*
  • Receptors, LDL / genetics*
  • Risk Assessment
  • Risk Factors
  • Young Adult

Substances

  • APOB protein, human
  • Apolipoprotein B-100
  • Biomarkers
  • Hydroxymethylglutaryl-CoA Reductase Inhibitors
  • LDLR protein, human
  • Lipids
  • Receptors, LDL
  • PCSK9 protein, human
  • Proprotein Convertase 9