Insights Into the Structure-Function Relationships of Dimeric C3d Fragments

Front Immunol. 2021 Aug 9:12:714055. doi: 10.3389/fimmu.2021.714055. eCollection 2021.

Abstract

Cleavage of C3 to C3a and C3b plays a central role in the generation of complement-mediated defences. Although the thioester-mediated surface deposition of C3b has been well-studied, fluid phase dimers of C3 fragments remain largely unexplored. Here we show C3 cleavage results in the spontaneous formation of C3b dimers and present the first X-ray crystal structure of a disulphide-linked human C3d dimer. Binding studies reveal these dimers are capable of crosslinking complement receptor 2 and preliminary cell-based analyses suggest they could modulate B cell activation to influence tolerogenic pathways. Altogether, insights into the physiologically-relevant functions of C3d(g) dimers gained from our findings will pave the way to enhancing our understanding surrounding the importance of complement in the fluid phase and could inform the design of novel therapies for immune system disorders in the future.

Keywords: B cell; C3d dimers; X-ray crystal and molecular structure; complement; tolerance.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Complement C3 / chemistry
  • Complement C3 / immunology
  • Complement C3d / chemistry*
  • Complement C3d / immunology
  • Humans
  • Lymphocyte Activation / immunology
  • Lymphocytes / immunology
  • Lymphocytes / metabolism
  • Models, Molecular*
  • Molecular Docking Simulation
  • Molecular Dynamics Simulation
  • Protein Conformation
  • Protein Multimerization*
  • Proteolysis
  • Recombinant Proteins / chemistry
  • Structure-Activity Relationship

Substances

  • Complement C3
  • Recombinant Proteins
  • Complement C3d