CD146 is a potential immunotarget for neuroblastoma

Cancer Sci. 2021 Nov;112(11):4617-4626. doi: 10.1111/cas.15124. Epub 2021 Sep 30.

Abstract

Neuroblastoma, the most common extracranial solid tumor of childhood, is thought to arise from neural crest-derived immature cells. The prognosis of patients with high-risk or recurrent/refractory neuroblastoma remains quite poor despite intensive multimodality therapy; therefore, novel therapeutic interventions are required. We examined the expression of a cell adhesion molecule CD146 (melanoma cell adhesion molecule [MCAM]) by neuroblastoma cell lines and in clinical samples and investigated the anti-tumor effects of CD146-targeting treatment for neuroblastoma cells both in vitro and in vivo. CD146 is expressed by 4 cell lines and by most of primary tumors at any stage. Short hairpin RNA-mediated knockdown of CD146, or treatment with an anti-CD146 polyclonal antibody, effectively inhibited growth of neuroblastoma cells both in vitro and in vivo, principally due to increased apoptosis via the focal adhesion kinase and/or nuclear factor-kappa B signaling pathway. Furthermore, the anti-CD146 polyclonal antibody markedly inhibited tumor growth in immunodeficient mice inoculated with primary neuroblastoma cells. In conclusion, CD146 represents a promising therapeutic target for neuroblastoma.

Keywords: CD146; antibody; apoptosis; focal adhesion kinase; neuroblastoma.

MeSH terms

  • Animals
  • Antibodies / therapeutic use*
  • Apoptosis
  • CD146 Antigen / antagonists & inhibitors*
  • CD146 Antigen / metabolism
  • Cell Line, Tumor
  • Cell Survival
  • Focal Adhesion Kinase 1 / metabolism
  • Focal Adhesion Protein-Tyrosine Kinases / metabolism
  • Gene Knockdown Techniques
  • Heterografts
  • Humans
  • Mice
  • Molecular Targeted Therapy / methods*
  • NF-kappa B / metabolism
  • Neoplasm Recurrence, Local
  • Neoplasm Transplantation
  • Neuroblastoma / metabolism
  • Neuroblastoma / pathology
  • Neuroblastoma / therapy*
  • Prognosis
  • RNA, Small Interfering / therapeutic use*
  • Signal Transduction
  • Spheroids, Cellular
  • Transduction, Genetic / methods

Substances

  • Antibodies
  • CD146 Antigen
  • NF-kappa B
  • RNA, Small Interfering
  • Focal Adhesion Kinase 1
  • Focal Adhesion Protein-Tyrosine Kinases
  • PTK2 protein, human