Virus-induced senescence is a driver and therapeutic target in COVID-19

Nature. 2021 Nov;599(7884):283-289. doi: 10.1038/s41586-021-03995-1. Epub 2021 Sep 13.

Abstract

Derailed cytokine and immune cell networks account for the organ damage and the clinical severity of COVID-19 (refs. 1-4). Here we show that SARS-CoV-2, like other viruses, evokes cellular senescence as a primary stress response in infected cells. Virus-induced senescence (VIS) is indistinguishable from other forms of cellular senescence and is accompanied by a senescence-associated secretory phenotype (SASP), which comprises pro-inflammatory cytokines, extracellular-matrix-active factors and pro-coagulatory mediators5-7. Patients with COVID-19 displayed markers of senescence in their airway mucosa in situ and increased serum levels of SASP factors. In vitro assays demonstrated macrophage activation with SASP-reminiscent secretion, complement lysis and SASP-amplifying secondary senescence of endothelial cells, which mirrored hallmark features of COVID-19 such as macrophage and neutrophil infiltration, endothelial damage and widespread thrombosis in affected lung tissue1,8,9. Moreover, supernatant from VIS cells, including SARS-CoV-2-induced senescence, induced neutrophil extracellular trap formation and activation of platelets and the clotting cascade. Senolytics such as navitoclax and a combination of dasatinib plus quercetin selectively eliminated VIS cells, mitigated COVID-19-reminiscent lung disease and reduced inflammation in SARS-CoV-2-infected hamsters and mice. Our findings mark VIS as a pathogenic trigger of COVID-19-related cytokine escalation and organ damage, and suggest that senolytic targeting of virus-infected cells is a treatment option against SARS-CoV-2 and perhaps other viral infections.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Aniline Compounds / pharmacology
  • Aniline Compounds / therapeutic use
  • Animals
  • COVID-19 / complications
  • COVID-19 / pathology*
  • COVID-19 / virology*
  • COVID-19 Drug Treatment*
  • Cell Line
  • Cellular Senescence / drug effects*
  • Cricetinae
  • Dasatinib / pharmacology
  • Dasatinib / therapeutic use
  • Disease Models, Animal
  • Female
  • Humans
  • Male
  • Mice
  • Molecular Targeted Therapy*
  • Quercetin / pharmacology
  • Quercetin / therapeutic use
  • SARS-CoV-2 / drug effects
  • SARS-CoV-2 / pathogenicity*
  • Sulfonamides / pharmacology
  • Sulfonamides / therapeutic use
  • Thrombosis / complications
  • Thrombosis / immunology
  • Thrombosis / metabolism

Substances

  • Aniline Compounds
  • Sulfonamides
  • Quercetin
  • Dasatinib
  • navitoclax