Disrupting cannabinoid receptor interacting protein 1 rescues cognitive flexibility in long-term estrogen-deprived female mice

Brain Res Bull. 2022 Apr:181:77-86. doi: 10.1016/j.brainresbull.2022.01.013. Epub 2022 Jan 29.

Abstract

Hormone therapy (HT) has failed to improve learning and memory in postmenopausal women according to recent clinical studies; however, the reason for failure of HT in improving cognitive performance is unknown. In our research, we found cognitive flexibility was improved by 17β-Estradiol (E2) in mice 1 week after ovariectomy (OVXST), but not in mice 3 months after ovariectomy (OVXLT). Isobaric tags for relative and absolute quantitation (iTRAQ) revealed increased cannabinoid receptor interacting protein 1 (CNRIP1) in E2-treated OVXLT mice compared with E2-treated OVXST mice. Adeno-associated virus 2/9 (AAV2/9) delivery of Cnrip1 short-hairpin small interfering RNA (Cnrip1-shRNA) rescued the impaired cognitive flexibility in E2 treated OVXLT mice. This effect is dependent on CB1 function, which could be blocked by AM251-a CB1 antagonist. Our results indicated a new method to increasing cognitive flexibility in women receiving HT by disrupting CNRIP1.

Keywords: Cannabinoid receptor interacting protein 1; Cognitive flexibility; Fear extinction; Hormone therapy; Medial prefrontal cortex.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cannabinoid Receptor Antagonists / pharmacology*
  • Carrier Proteins / drug effects*
  • Carrier Proteins / metabolism*
  • Cognitive Dysfunction / drug therapy*
  • Cognitive Dysfunction / metabolism*
  • Disease Models, Animal
  • Estradiol / pharmacology*
  • Female
  • Hormone Replacement Therapy*
  • Mice
  • Ovariectomy
  • Piperidines / pharmacology
  • Postmenopause
  • Prefrontal Cortex / drug effects*
  • Pyrazoles / pharmacology
  • RNA, Small Interfering
  • Receptor, Cannabinoid, CB1 / antagonists & inhibitors

Substances

  • CRIP1a protein, mouse
  • Cannabinoid Receptor Antagonists
  • Carrier Proteins
  • Piperidines
  • Pyrazoles
  • RNA, Small Interfering
  • Receptor, Cannabinoid, CB1
  • AM 251
  • Estradiol