Enzyme active sites: Identification and prediction of function using computational chemistry

Curr Opin Struct Biol. 2022 Jun:74:102384. doi: 10.1016/j.sbi.2022.102384. Epub 2022 May 6.

Abstract

Understanding the biochemically active amino acids in proteins is a key factor to improve the knowledge of how enzymes work, to predict the function of newly discovered protein structures of unknown function, and to establish design principles for enzyme engineering. Here, we explore recently reported computational chemistry-based methods for the prediction of active amino acids in protein 3D structures, including biochemically important distal residues, and their implications for functional genomics, for enzyme design, and for enhancing understanding of the function of enzymes.

Publication types

  • Review
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Amino Acids / chemistry
  • Catalytic Domain
  • Computational Biology / methods
  • Computational Chemistry*
  • Enzymes / chemistry
  • Proteins* / chemistry

Substances

  • Amino Acids
  • Enzymes
  • Proteins