Rituximab abrogates aquaporin-4-specific germinal center activity in patients with neuromyelitis optica spectrum disorders

Proc Natl Acad Sci U S A. 2022 Jun 14;119(24):e2121804119. doi: 10.1073/pnas.2121804119. Epub 2022 Jun 6.

Abstract

Neuromyelitis optica spectrum disorders (NMOSDs) are caused by immunoglobulin G (IgG) autoantibodies directed against the water channel aquaporin-4 (AQP4). In NMOSDs, discrete clinical relapses lead to disability and are robustly prevented by the anti-CD20 therapeutic rituximab; however, its mechanism of action in autoantibody-mediated disorders remains poorly understood. We hypothesized that AQP4-IgG production in germinal centers (GCs) was a core feature of NMOSDs and could be terminated by rituximab. To investigate this directly, deep cervical lymph node (dCLN) aspirates (n = 36) and blood (n = 406) were studied in a total of 63 NMOSD patients. Clinical relapses were associated with AQP4-IgM generation or shifts in AQP4-IgG subclasses (odds ratio = 6.0; range of 3.3 to 10.8; P < 0.0001), features consistent with GC activity. From seven dCLN aspirates of patients not administered rituximab, AQP4-IgGs were detected alongside specific intranodal synthesis of AQP4-IgG. AQP4-reactive B cells were isolated from unmutated naive and mutated memory populations in both blood and dCLNs. After rituximab administration, fewer clinical relapses (annual relapse rate of 0.79 to 0; P < 0.001) were accompanied by marked reductions in both AQP4-IgG (fourfold; P = 0.004) and intranodal B cells (430-fold; P < 0.0001) from 11 dCLNs. Our findings implicate ongoing GC activity as a rituximab-sensitive driver of AQP4 antibody production. They may explain rituximab’s clinical efficacy in several autoantibody-mediated diseases and highlight the potential value of direct GC measurements across autoimmune conditions.

Keywords: aquaporin; autoimmunity; cervical lymph nodes; neuromyelitis optica; rituximab.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aquaporin 4* / drug effects
  • Aquaporin 4* / metabolism
  • Autoantibodies
  • Germinal Center* / pathology
  • Humans
  • Immunologic Factors* / pharmacology
  • Immunologic Factors* / therapeutic use
  • Lymph Nodes / metabolism
  • Neuromyelitis Optica* / drug therapy
  • Rituximab* / pharmacology
  • Rituximab* / therapeutic use

Substances

  • Aquaporin 4
  • Autoantibodies
  • Immunologic Factors
  • Rituximab