D3 Receptors and PET Imaging

Curr Top Behav Neurosci. 2023:60:251-275. doi: 10.1007/7854_2022_374.

Abstract

This chapter encapsulates a short introduction to positron emission tomography (PET) imaging and the information gained by using this technology to detect changes of the dopamine 3 receptor (D3R) at the molecular level in vivo. We will discuss available D3R radiotracers, emphasizing [11C]PHNO. The focus, however, will be on PET findings in conditions including substance abuse, obesity, traumatic brain injury, schizophrenia, Parkinson's disease, and aging. Finally, there is a discussion about progress in producing next-generation selective D3R radiotracers.

Keywords: D3; Dopamine; Humans; PET imaging.

MeSH terms

  • Brain / diagnostic imaging
  • Brain / metabolism
  • Humans
  • Oxazines
  • Positron-Emission Tomography / methods
  • Receptors, Dopamine D2* / metabolism
  • Receptors, Dopamine D3 / metabolism
  • Schizophrenia*

Substances

  • Receptors, Dopamine D2
  • Receptors, Dopamine D3
  • Oxazines