Ketamine triggers rapid antidepressant effects by modulating synaptic plasticity in a new depressive-like mouse model based on astrocyte glutamate transporter GLT-1 knockdown in infralimbic cortex

Rev Psiquiatr Salud Ment (Engl Ed). 2022 Apr-Jun;15(2):94-100. doi: 10.1016/j.rpsmen.2022.06.008.

Abstract

Objective: Recently, we reported on a new MDD-like mouse model based on a regionally selective knockdown of astroglial glutamate transporters, GLAST/GLT-1, in infralimbic cortex (IL) which evokes widespread changes in mouse brain associated with the typical alterations found in MDD patients. To further characterize this new MDD-like mouse model, here we examine some transcriptional elements of glutamatergic/GABAergic neurotransmission and neuroplasticity in forebrain regions in the GLT-1 knockdown mice. Furthermore, we assess the acute ketamine effects on these transcriptional processes.

Material and methods: We used a small interfering RNA (siRNA) pool targeting GLT-1 mRNA to disrupt the GLT-1 transcription in mouse IL. Histological assays were performed to examine postsynaptic density protein-95 (PSD95), neuritin (NRN), glutamine acid descarboxilase-65 (GAD65), and GLT-1 mRNA expression in IL and hippocampus.

Results: Knockdown of GLT-1 in mouse IL leads to decreased expression of PSD95 and NRN neuroplasticity mRNAs in IL and hippocampus, which was reversed by an acute dose of ketamine antidepressant. Likewise, a single dose of ketamine also increased the mRNA levels of GAD65 and GLT-1 in IL of GLT-1 knockdown mice, reaching the basal values of control mice.

Conclusions: The glutamatergic neuronal hyperactivity and deficits in the GABA system resulting from siRNA-induced astroglial glutamate transporter knockdown in IL can compromise the integrity/plasticity of neurocircuits affected in MDD. Suitable depressive-like animal models to address the neurobiological changes in MDD are an unmet need and the development of the GLAST/GLT-1 knockdown mouse model may represent a better option to understand the rapid-acting antidepressant effects of ketamine.

Keywords: Astrocitos; Astrocytes; Corteza infralímbica; Depresión; Depression; Infralimbic cortex; Ketamina; Ketamine; PSD95.

MeSH terms

  • Amino Acid Transport System X-AG / metabolism
  • Animals
  • Antidepressive Agents / pharmacology
  • Antidepressive Agents / therapeutic use
  • Astrocytes* / metabolism
  • Depression / genetics
  • Depression / metabolism
  • Excitatory Amino Acid Transporter 2 / drug effects
  • Excitatory Amino Acid Transporter 2 / genetics
  • Humans
  • Ketamine* / metabolism
  • Ketamine* / pharmacology
  • Ketamine* / therapeutic use
  • Mice
  • Neuronal Plasticity* / drug effects
  • Neuronal Plasticity* / genetics
  • RNA, Messenger / metabolism
  • RNA, Small Interfering / metabolism

Substances

  • Amino Acid Transport System X-AG
  • Antidepressive Agents
  • Excitatory Amino Acid Transporter 2
  • RNA, Messenger
  • RNA, Small Interfering
  • Slc1a2 protein, mouse
  • Ketamine