FGFR3-TACCs3 Fusions and Their Clinical Relevance in Human Glioblastoma

Int J Mol Sci. 2022 Aug 4;23(15):8675. doi: 10.3390/ijms23158675.

Abstract

Oncogenic fusion genes have emerged as successful targets in several malignancies, such as chronic myeloid leukemia and lung cancer. Fusion of the fibroblast growth receptor 3 and the transforming acidic coiled coil containing protein-FGFR3-TACC3 fusion-is prevalent in 3-4% of human glioblastoma. The fusion protein leads to the constitutively activated kinase signaling of FGFR3 and thereby promotes cell proliferation and tumor progression. The subgroup of FGFR3-TACC3 fusion-positive glioblastomas presents with recurrent clinical and histomolecular characteristics, defining a distinctive subtype of IDH-wildtype glioblastoma. This review aims to provide an overview of the available literature on FGFR3-TACC3 fusions in glioblastoma and possible implications for actual clinical practice.

Keywords: FGFR; FGFR3-TACC3; TACC; glioblastoma; molecular diagnostics; molecular signaling; oncogenic fusion; tyrosine kinase receptors.

Publication types

  • Review

MeSH terms

  • Gene Fusion
  • Glioblastoma* / genetics
  • Humans
  • Lung Neoplasms*
  • Microtubule-Associated Proteins / metabolism
  • Oncogene Fusion
  • Receptor, Fibroblast Growth Factor, Type 3 / genetics
  • Receptor, Fibroblast Growth Factor, Type 3 / metabolism

Substances

  • Microtubule-Associated Proteins
  • TACC3 protein, human
  • FGFR3 protein, human
  • Receptor, Fibroblast Growth Factor, Type 3

Grants and funding

This research received no external funding.