BMP4 and Gremlin 1 regulate hepatic cell senescence during clinical progression of NAFLD/NASH

Nat Metab. 2022 Aug;4(8):1007-1021. doi: 10.1038/s42255-022-00620-x. Epub 2022 Aug 22.

Abstract

The role of hepatic cell senescence in human non-alcoholic fatty liver disease (NAFLD) and non-alcoholic steatohepatitis (NASH) is not well understood. To examine this, we performed liver biopsies and extensive characterization of 58 individuals with or without NAFLD/NASH. Here, we show that hepatic cell senescence is strongly related to NAFLD/NASH severity, and machine learning analysis identified senescence markers, the BMP4 inhibitor Gremlin 1 in liver and visceral fat, and the amount of visceral adipose tissue as strong predictors. Studies in liver cell spheroids made from human stellate and hepatocyte cells show BMP4 to be anti-senescent, anti-steatotic, anti-inflammatory and anti-fibrotic, whereas Gremlin 1, which is particularly highly expressed in visceral fat in humans, is pro-senescent and antagonistic to BMP4. Both senescence and anti-senescence factors target the YAP/TAZ pathway, making this a likely regulator of senescence and its effects. We conclude that senescence is an important driver of human NAFLD/NASH and that BMP4 and Gremlin 1 are novel therapeutic targets.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, N.I.H., Extramural

MeSH terms

  • Bone Morphogenetic Protein 4 / metabolism
  • Cellular Senescence
  • Hepatocytes / metabolism
  • Humans
  • Intercellular Signaling Peptides and Proteins / metabolism*
  • Intra-Abdominal Fat / metabolism
  • Non-alcoholic Fatty Liver Disease* / metabolism

Substances

  • BMP4 protein, human
  • Bone Morphogenetic Protein 4
  • GREM1 protein, human
  • Intercellular Signaling Peptides and Proteins