Upregulated miR-194-5p suppresses retinal microvascular endothelial cell dysfunction and mitigates the symptoms of hypertensive retinopathy in mice by targeting SOX17 and VEGF signaling

Cell Cycle. 2023 Feb;22(3):331-346. doi: 10.1080/15384101.2022.2119514. Epub 2022 Oct 5.

Abstract

Background: Hypertensive retinopathy (HR) is a retinal disease that may lead to vision loss and blindness. Sex-determining region Y (SRY)-box (SOX) family transcription factors have been reported to be involved in HR development. In this study, the role and upstream mechanism of SRY-box transcription factor 17 (SOX17) in HR pathogenesis were investigated.

Methods: SOX17 and miR-194-5p levels in Angiotensin II (Ang II)-stimulated human retinal microvascular endothelial cells (HRMECs) and retinas of mice were detected by RT-qPCR. SOX17 protein level as well as levels of tight junction proteins and vascular endothelial growth factor (VEGF) signaling-associated proteins were quantified by western blotting. Tube formation assays were performed to evaluate angiogenesis in HRMECs. The structure of mouse retinal tissues was observed by H&E staining. The interaction between miR-194-5p and SOX17 was confirmed by a luciferase reporter assay.

Results: SOX17 was upregulated in HRMECs treated with Ang II. SOX17 knockdown inhibited angiogenesis in Ang II-stimulated HRMECs and increased tight junction protein levels. Mechanically, SOX17 was targeted by miR-194-5p. Moreover, miR-194-5p upregulation restrained angiogenesis and increased tight junction protein levels in Ang II-treated HRMECs, and the effect was reversed by SOX17 overexpression. MiR-194-5p elevation inactivated VEGF signaling via targeting SOX17. miR-194-5p alleviated pathological symptoms of HR in Ang II-treated mice, and its expression was negatively correlated with SOX17 expression in the retinas of model mice.

Conclusions: MiR-194-5p upregulation suppressed Ang II-stimulated HRMEC dysfunction and mitigates the symptoms of HR in mice by regulating the SOX17/VEGF signaling.

Keywords: HRMEC; Hypertensive retinopathy; SOX17; VEGF signaling; angiogenesis; miR-194-5p.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cell Proliferation
  • Endothelial Cells / metabolism
  • HMGB Proteins / metabolism
  • HMGB Proteins / pharmacology
  • Humans
  • Hypertensive Retinopathy* / metabolism
  • Hypertensive Retinopathy* / pathology
  • Mice
  • MicroRNAs* / genetics
  • MicroRNAs* / metabolism
  • SOXF Transcription Factors / genetics
  • SOXF Transcription Factors / metabolism
  • SOXF Transcription Factors / pharmacology
  • Tight Junction Proteins / metabolism
  • Vascular Endothelial Growth Factor A / metabolism
  • Vascular Endothelial Growth Factors / metabolism
  • Vascular Endothelial Growth Factors / pharmacology

Substances

  • Vascular Endothelial Growth Factor A
  • MicroRNAs
  • Vascular Endothelial Growth Factors
  • Tight Junction Proteins
  • SOX17 protein, human
  • SOXF Transcription Factors
  • MIRN194 microRNA, human
  • Sox17 protein, mouse
  • HMGB Proteins

Grants and funding

The research was supported by Research Fund of Anhui Medical University (grant no: 2020xkj202)