Exceptional response to neoadjuvant targeted therapy with the selective RET inhibitor selpercatinib in RET-fusion-associated sarcoma

J Cancer Res Clin Oncol. 2023 Aug;149(9):5493-5496. doi: 10.1007/s00432-022-04496-y. Epub 2022 Dec 5.

Abstract

With the increasing use of next-generation sequencing, highly effective targeted therapies have been emerging as treatment options for several cancer types. Recurrent gene-fusions have been recognized in sarcomas; however, options for targeted therapy remain scarce. Here, we describe a case of a sarcoma, associated with a RET::TRIM33-fusion gene with an exceptional response to a neoadjuvant therapy with the selective RET inhibitor selpercatinib. Resected tumor revealed subtotal histopathologic response. This is the first report of successful targeted therapy with selpercatinib in RET-fusion-associated sarcomas. As new targeted therapies are under development, similar treatment options may become available for sarcoma patients.

Keywords: RET-fusion; Sarcoma; Selpercatinib; TRIM33; Targeted therapy.

Publication types

  • Case Reports

MeSH terms

  • Humans
  • Lung Neoplasms*
  • Neoadjuvant Therapy
  • Protein Kinase Inhibitors / therapeutic use
  • Proto-Oncogene Proteins c-ret / genetics
  • Pyrazoles
  • Pyridines
  • Sarcoma* / drug therapy
  • Sarcoma* / genetics
  • Soft Tissue Neoplasms*
  • Transcription Factors

Substances

  • selpercatinib
  • Pyrazoles
  • Pyridines
  • Protein Kinase Inhibitors
  • RET protein, human
  • Proto-Oncogene Proteins c-ret
  • TRIM33 protein, human
  • Transcription Factors