[Pharmacokinetics and metabolism of cyclosporin; drug interactions]

Nephrologie. 1987;8(3):135-41.
[Article in French]

Abstract

The pharmacokinetic properties of cyclosporine and mainly its absorption and hepatic elimination can vary in each patient in relation to the subject's individual characteristics (inter-subject variability), as well as in an individual patient during his treatment because of clinical episodes or drug interactions (intra-subject variabilities). Therefore, it appears compulsory to follow regularly cyclosporine blood levels or even to characterise each subject following a dose-test during the initiation of treatment, in order to adapt an individual posology aiming to minimise as far as possible the risk of nephrotoxicity.

Publication types

  • English Abstract

MeSH terms

  • Administration, Oral
  • Animals
  • Biotransformation
  • Cyclosporins / administration & dosage
  • Cyclosporins / antagonists & inhibitors
  • Cyclosporins / pharmacokinetics*
  • Dogs
  • Drug Interactions
  • Erythromycin / pharmacology
  • Humans
  • Injections, Intravenous
  • Ketoconazole / pharmacology
  • Liver / metabolism
  • Methylprednisolone / pharmacology
  • Rabbits
  • Rats
  • Tissue Distribution

Substances

  • Cyclosporins
  • Erythromycin
  • Ketoconazole
  • Methylprednisolone