ATM suppresses c-Myc overexpression in the mammary epithelium in response to estrogen

Cell Rep. 2023 Jan 31;42(1):111909. doi: 10.1016/j.celrep.2022.111909. Epub 2022 Dec 30.

Abstract

ATM gene mutation carriers are predisposed to estrogen-receptor-positive breast cancer (BC). ATM prevents BC oncogenesis by activating p53 in every cell; however, much remains unknown about tissue-specific oncogenesis after ATM loss. Here, we report that ATM controls the early transcriptional response to estrogens. This response depends on topoisomerase II (TOP2), which generates TOP2-DNA double-strand break (DSB) complexes and rejoins the breaks. When TOP2-mediated ligation fails, ATM facilitates DSB repair. After estrogen exposure, TOP2-dependent DSBs arise at the c-MYC enhancer in human BC cells, and their defective repair changes the activation profile of enhancers and induces the overexpression of many genes, including the c-MYC oncogene. CRISPR/Cas9 cleavage at the enhancer also causes c-MYC overexpression, indicating that this DSB causes c-MYC overexpression. Estrogen treatment induced c-Myc protein overexpression in mammary epithelial cells of ATM-deficient mice. In conclusion, ATM suppresses the c-Myc-driven proliferative effects of estrogens, possibly explaining such tissue-specific oncogenesis.

Keywords: CP: Cancer; CP: Cell biology; DNA double-strand break repair; ataxia-telangiectasia (ATM); breast cancer; c-MYC; enhancer; estradiol; topoisomerase II.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, N.I.H., Extramural
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Animals
  • Ataxia Telangiectasia Mutated Proteins / metabolism
  • Carcinogenesis / genetics
  • Cell Cycle Proteins / metabolism
  • DNA Breaks, Double-Stranded*
  • DNA Repair
  • Epithelium / metabolism
  • Estrogens / pharmacology
  • Genes, myc*
  • Humans
  • Mice

Substances

  • Ataxia Telangiectasia Mutated Proteins
  • Estrogens
  • Cell Cycle Proteins
  • ATM protein, human