Hypoxia-Inducible Factor-2alpha Affects the MEK/ERK Signaling Pathway via Primary Cilia in Connection with the Intraflagellar Transport Protein 88 Homolog

Mol Cell Biol. 2023;43(4):174-183. doi: 10.1080/10985549.2023.2198931. Epub 2023 Apr 19.

Abstract

The ability of cells to communicate with their surrounding is a prerequisite for essential processes such as proliferation, apoptosis, migration, and differentiation. To this purpose, primary cilia serve as antennae-like structures on the surface of most mammalian cell types. Cilia allow signaling via hedgehog, Wnt or TGF-beta pathways. Their length, in part controlled by the activity of intraflagellar transport (IFT), is a parameter for adequate function of primary cilia. Here we show, in murine neuronal cells, that intraflagellar transport protein 88 homolog (IFT88) directly interacts with the hypoxia-inducible factor-2α (HIF-2α), hitherto known as an oxygen-regulated transcription factor. Furthermore, HIF-2α accumulates in the ciliary axoneme and promotes ciliary elongation under hypoxia. Loss of HIF-2α affected ciliary signaling in neuronal cells by decreasing transcription of Mek1/2 and Erk1/2. Targets of the MEK/ERK signaling pathway, such as Fos and Jun, were significantly decreased. Our results suggest that HIF-2α influences ciliary signaling by interacting with IFT88 under hypoxic conditions. This implies an unexpected and far more extensive function of HIF-2α than described before.

Keywords: HIF-2; IFT88; MEK/ERK signaling; primary cilia.

MeSH terms

  • Animals
  • Basic Helix-Loop-Helix Transcription Factors* / metabolism
  • Carrier Proteins / metabolism
  • Cilia* / metabolism
  • Hypoxia
  • Hypoxia-Inducible Factor 1, alpha Subunit / metabolism
  • Mammals / metabolism
  • Mice
  • Mitogen-Activated Protein Kinase Kinases / metabolism
  • Signal Transduction
  • Transcription Factors / metabolism

Substances

  • Basic Helix-Loop-Helix Transcription Factors
  • Transcription Factors
  • Carrier Proteins
  • Mitogen-Activated Protein Kinase Kinases
  • Hypoxia-Inducible Factor 1, alpha Subunit

Associated data

  • figshare/10.6084/m9.figshare.21975563.v1