Tolerance to ethanol and cross-tolerance to pentobarbital and barbital

Pharmacol Biochem Behav. 1986 Apr;24(4):801-7. doi: 10.1016/0091-3057(86)90414-4.

Abstract

A chronic regimen of ethanol by intubation, which produced clear tolerance to ethanol-induced hypothermia, ataxia and narcosis, produced only a marginal degree of cross-tolerance to these effects of pentobarbital. The lack of appreciable cross-tolerance to pentobarbital-induced hypothermia and ataxia was also observed over a wide range of test doses. However, cross-tolerance to barbital was observed after chronic treatment with ethanol. Increased rate of drug biotransformation did not contribute significantly to the observed tolerance and cross-tolerance. The difference in the extent of cross-tolerance between ethanol and the two barbiturates is consistent with the hypothesis that there is a degree of specificity in the sites of action of ethanol and other sedative-hypnotic drugs.

Publication types

  • Comparative Study

MeSH terms

  • Animals
  • Barbital / pharmacology*
  • Barbiturates / pharmacology*
  • Body Temperature / drug effects
  • Dose-Response Relationship, Drug
  • Drug Tolerance
  • Ethanol / pharmacology*
  • Male
  • Motor Activity / drug effects
  • Pentobarbital / pharmacology*
  • Rats
  • Rats, Inbred Strains
  • Sleep / drug effects

Substances

  • Barbiturates
  • Ethanol
  • Barbital
  • Pentobarbital