The induced and intrinsic resistance of Escherichia coli to sanguinarine is mediated by AcrB efflux pump

Microbiol Spectr. 2024 Jan 11;12(1):e0323723. doi: 10.1128/spectrum.03237-23. Epub 2023 Dec 1.

Abstract

The use of plant extracts is increasing as an alternative to synthetic compounds, especially antibiotics. However, there is no sufficient knowledge on the mechanisms and potential risks of antibiotic resistance induced by these phytochemicals. In the present study, we found that stable drug resistant mutants of E. coli emerged after repetitive exposure to sanguinarine and demonstrated that the AcrB efflux pump contributed to the emerging of induced and intrinsic resistance of E. coli to this phytochemical. Our results offered some insights into comprehending and preventing the onset of drug-resistant strains when utilizing products containing sanguinarine.

Keywords: AcrB; Escherichia coli; antibiotic alternatives; antimicrobial resistance; efflux pump; sanguinarine.

MeSH terms

  • Anti-Bacterial Agents / chemistry
  • Anti-Bacterial Agents / pharmacology
  • Benzophenanthridines*
  • Drug Resistance, Multiple, Bacterial
  • Escherichia coli Proteins* / genetics
  • Escherichia coli Proteins* / metabolism
  • Escherichia coli* / genetics
  • Escherichia coli* / metabolism
  • Isoquinolines*
  • Microbial Sensitivity Tests
  • Multidrug Resistance-Associated Proteins / genetics

Substances

  • Escherichia coli Proteins
  • sanguinarine
  • Anti-Bacterial Agents
  • AcrB protein, E coli
  • Multidrug Resistance-Associated Proteins
  • Isoquinolines
  • Benzophenanthridines