Rapid Initiation of Antiretroviral Therapy With Coformulated Bictegravir, Emtricitabine, and Tenofovir Alafenamide Versus Efavirenz, Lamivudine, and Tenofovir Disoproxil Fumarate in HIV-Positive Men Who Have Sex With Men in China: Week 48 Results of the Multicenter, Randomized Clinical Trial

Clin Infect Dis. 2024 Jul 19;79(1):169-176. doi: 10.1093/cid/ciae012.

Abstract

Background: Most international treatment guidelines recommend rapid initiation of antiretroviral therapy (ART) for people newly diagnosed with human immunodeficiency virus (HIV)-1 infection, but experiences with rapid ART initiation remain limited in China. We aimed to evaluate the efficacy and safety of efavirenz (400 mg) plus lamivudine and tenofovir disoproxil fumarate (EFV + 3TC + TDF) versus coformulated bictegravir, emtricitabine, and tenofovir alafenamide (BIC/FTC/TAF) in rapid ART initiation among men who have sex with men (MSM) who have been diagnosed with HIV.

Methods: This multicenter, open-label, randomized clinical trial enrolled MSM aged ≥18 years to start ART within 14 days of confirmed HIV diagnosis. The participants were randomly assigned in a 1:1 ratio to receive EFV (400 mg) + 3TC + TDF or BIC/FTC/TAF. The primary end point was viral suppression (<50 copies/mL) at 48 weeks per US Food and Drug Administration Snapshot analysis.

Results: Between March 2021 and July 2022, 300 participants were enrolled; 154 were assigned to receive EFV + 3TC + TDF (EFV group) and 146 BIC/FTC/TAF (BIC group). At week 48, 118 (79.2%) and 140 (95.9%) participants in the EFV and BIC group, respectively, were retained in care with viral suppression, and 24 (16.1%) and 1 (0.7%) participant in the EFV and BIC group (P < .001), respectively, discontinued treatment because of adverse effects, death, or lost to follow-up. The median increase of CD4 count was 181 and 223 cells/μL (P = .020), respectively, for the EFV and BIC group, at week 48. The overall incidence of adverse effects was significantly higher for the EFV group (65.8% vs 37.7%, P < .001).

Conclusions: BIC/FTC/TAF was more efficacious and safer than EFV (400 mg) + 3TC + TDF for rapid ART initiation among HIV-positive MSM in China.

Keywords: care cascade; integrase strand-transfer inhibitor; non-nucleoside reverse-transcriptase inhibitor; treatment retention; treatment-as-prevention.

Publication types

  • Randomized Controlled Trial
  • Multicenter Study

MeSH terms

  • Adult
  • Alanine / therapeutic use
  • Alkynes* / therapeutic use
  • Amides
  • Anti-HIV Agents* / administration & dosage
  • Anti-HIV Agents* / adverse effects
  • Anti-HIV Agents* / therapeutic use
  • Antiretroviral Therapy, Highly Active / methods
  • Benzoxazines* / therapeutic use
  • CD4 Lymphocyte Count
  • China
  • Cyclopropanes* / therapeutic use
  • Dioxolanes / administration & dosage
  • Dioxolanes / therapeutic use
  • Drug Combinations
  • Emtricitabine* / administration & dosage
  • Emtricitabine* / therapeutic use
  • HIV Infections* / drug therapy
  • HIV-1 / drug effects
  • Heterocyclic Compounds, 3-Ring / administration & dosage
  • Heterocyclic Compounds, 3-Ring / adverse effects
  • Heterocyclic Compounds, 3-Ring / therapeutic use
  • Heterocyclic Compounds, 4 or More Rings / administration & dosage
  • Heterocyclic Compounds, 4 or More Rings / adverse effects
  • Heterocyclic Compounds, 4 or More Rings / therapeutic use
  • Homosexuality, Male*
  • Humans
  • Lamivudine* / administration & dosage
  • Lamivudine* / adverse effects
  • Lamivudine* / therapeutic use
  • Male
  • Middle Aged
  • Piperazines / therapeutic use
  • Pyridones
  • Tenofovir* / analogs & derivatives
  • Tenofovir* / therapeutic use
  • Viral Load
  • Young Adult

Substances

  • Tenofovir
  • Emtricitabine
  • Cyclopropanes
  • Anti-HIV Agents
  • Alkynes
  • Lamivudine
  • Benzoxazines
  • efavirenz
  • Alanine
  • Heterocyclic Compounds, 4 or More Rings
  • bictegravir
  • tenofovir alafenamide
  • Dioxolanes
  • Heterocyclic Compounds, 3-Ring
  • Piperazines
  • Drug Combinations
  • Amides
  • Pyridones