Kinetics of iodomethylated hexadecanoic acid metabolism in the rat myocardium: influence of the number and the position of methyl radicals

Int J Nucl Med Biol. 1985;12(5):363-7.

Abstract

The methyl-branched fatty acids, if radioiodine labelled in alpha position, are potentially adapted to a selective study of FA myocardial uptake. To determine the position and the number of methyl radicals that are necessary to obtain a maximal uptake and a minimal degradation, we measured time-activity evolution of isolated and perfused rat hearts after an injection of iodinated fatty acids which are mono- or dimethylated in alpha or beta position. Except for dimethyl fatty acid, the uptake is similar for all fatty acids studied to that of the straight chain analogue; beta mono- or dimethyl fatty acids seem best adapted to a study of the uptake because alpha monomethyl fatty acids undergo a metabolic degradation and alpha mono- and dimethyl fatty acids induce ventricular fibrillations.

MeSH terms

  • Animals
  • In Vitro Techniques
  • Iodine Radioisotopes
  • Kinetics
  • Male
  • Methylation
  • Myocardium / metabolism*
  • Palmitic Acids / metabolism*
  • Rats
  • Rats, Inbred Strains
  • Structure-Activity Relationship
  • Ventricular Fibrillation

Substances

  • Iodine Radioisotopes
  • Palmitic Acids