Crebinostat facilitates memory formation

Biochem Biophys Res Commun. 2024 May 28:710:149872. doi: 10.1016/j.bbrc.2024.149872. Epub 2024 Apr 4.

Abstract

Protein modifications importantly contribute to memory formation. Protein acetylation is a post-translational modification of proteins that regulates memory formation. Acetylation level is determined by the relative activities of acetylases and deacetylases. Crebinostat is a histone deacetylase inhibitor. Here we show that in an object recognition task, crebinostat facilitates memory formation by a weak training. Further, this compound enhances acetylation of α-tubulin, and reduces the level of histone deacetylase 6, an α-tubulin deacetylase. The results suggest that enhanced acetylation of α-tubulin by crebinostat contributes to its facilitatory effect on memory formation.

Keywords: Acetylation; HDAC6; Memory; Object recognition task; α-tubulin.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acetylation
  • Biphenyl Compounds
  • Histone Deacetylase 6 / metabolism
  • Histone Deacetylase Inhibitors / pharmacology
  • Histone Deacetylases* / metabolism
  • Hydrazines
  • Tubulin* / metabolism

Substances

  • Tubulin
  • Histone Deacetylases
  • (7-(2-((1,1'-biphenyl)-4-ylmethylene)hydrazinyl)-N-hydroxy-7-oxoheptanamide)
  • Histone Deacetylase 6
  • Biphenyl Compounds
  • Hydrazines
  • Histone Deacetylase Inhibitors