Artificial fluorescent sensor reveals pre-synaptic NMDA receptors switch cholecystokinin release and LTP in the hippocampus

J Neurochem. 2024 Sep;168(9):2621-2639. doi: 10.1111/jnc.16128. Epub 2024 May 15.

Abstract

Cholecystokinin (CCK) has been confirmed to be essential in NMDA-dependent long-term potentiation (LTP) at mouse cortical synapses. This paper has proven that CCK is necessary for LTP induced by high-frequency stimulation of mouse hippocampal synapses projected from the entorhinal cortex. We show that the subunit of the axonal NMDA receptor dominant modulates the activity-induced LTP by triggering pre-synaptic CCK release. A functional pre-synaptic NMDA receptor is required to induce LTP mediated by the axonal Ca2+ elevation and CCK exocytosis at CCK-specific neurons. Genetic depletion of the GluN1 subunit of NMDA receptors on CCK neurons, which projected from the entorhinal cortex largely abolished the axonal Ca2+ elevation and disturbed the secretion of CCK in hippocampus. These results demonstrate that activity-induced LTP at the hippocampal synapse is CCK-dependent, and CCK secretion from the axonal terminal is modulated by pre-synaptic NMDA receptors.

Keywords: Ca2+; NMDA receptor; cholecystokinin; hippocampus; long‐term potentiation.

MeSH terms

  • Animals
  • Cholecystokinin* / metabolism
  • Hippocampus* / metabolism
  • Long-Term Potentiation* / physiology
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Presynaptic Terminals / metabolism
  • Receptors, N-Methyl-D-Aspartate* / metabolism
  • Synapses / metabolism

Substances

  • Receptors, N-Methyl-D-Aspartate
  • Cholecystokinin