Evaluation of the in-vitro antibacterial activity of Sch 34343

J Antimicrob Chemother. 1985 Jun:15 Suppl C:39-56. doi: 10.1093/jac/15.suppl_c.39.

Abstract

The in-vitro activity (as measured by geometric mean MICs, mg/l) of Sch 34343 against aerobic and anaerobic bacteria was compared with that of 14 other selected beta-lactam antibiotics including aztreonam, latamoxef (moxalactam), ceftazidime and imipenem. Sch 34343 had good activity (less than 2 mg/l) against most Gram-negative aerobic bacteria whether or not they contained high levels of plasmid-mediated or chromosomally-mediated beta-lactamases. It was slightly less potent against strains of Morganella and Serratia (less than 4 mg/l) and inactive against Pseudomonas (greater than 64 mg/l). A very small inoculum effect was observed against strains containing beta-lactamases indicating stability. Unlike the third-generation cephalosporins, Sch 34343 had excellent activity (less than or equal to 0.18 mg/l) against staphylococci, comparable to that of imipenem and ampicillin. While Sch 34343 had equally good potency (0.17 mg/l) against penicillinase-positive staphylococci, it was inactive against methicillin-resistant staphylococci (greater than or equal to 35 mg/l). Sch 34343 also had good activity against streptococci. The most unusual aspect of the in-vitro activity was its activity against Bacteroides (including Bact. fragilis) and other anaerobes. Sch 34343 had mean MICs less than or equal to mg/l for all Bacteroides and Clostridium spp. tested except CI. difficile (3.4 mg/l).

MeSH terms

  • Anti-Bacterial Agents / blood
  • Anti-Bacterial Agents / pharmacology*
  • Bacteria / drug effects*
  • Bacteria / enzymology
  • Bacteria, Aerobic / drug effects
  • Bacteria, Anaerobic / drug effects
  • Blood Proteins / metabolism
  • Gram-Negative Bacteria / drug effects
  • Gram-Negative Bacteria / enzymology
  • Gram-Positive Bacteria / drug effects
  • Haemophilus / drug effects
  • Lactams*
  • Microbial Sensitivity Tests
  • Neisseria / drug effects
  • Protein Binding
  • Streptococcus / drug effects
  • beta-Lactamases / metabolism
  • beta-Lactams*

Substances

  • Anti-Bacterial Agents
  • Blood Proteins
  • Lactams
  • beta-Lactams
  • Sch 34343
  • beta-Lactamases