Psychedelic 25H-NBOMe attenuates post-sepsis depression in rats

Neurosci Lett. 2024 Jun 21:834:137845. doi: 10.1016/j.neulet.2024.137845. Epub 2024 May 29.

Abstract

Sepsis-associated encephalopathy, which manifests in severe cognitive and depressive symptoms, is directly linked to neuroinflammation. Our study investigates the efficacy of 25H-NBOMe, a phenethylamine, in alleviating these symptoms, potentially offering an innovative treatment for post-sepsis depression. Wistar rats, weighing between 250-300 g, were subjected to cecal ligation and puncture (CLP) surgery to induce sepsis. Depressive-like behaviors were assessed using the forced swim test (FST) on either day 7 or 14 post-surgery, to establish the presence of depressive symptoms. The impact of 25H-NBOMe treatment was then evaluated, focusing on the head-twitch response (HTR), performance in the FST, and GFAP expression in the prefrontal cortex. Treatment with 25H-NBOMe resulted in significant behavioral changes, demonstrated by decreased immobility and increased swimming times in the FST, along with a rise in the HTR. These outcomes indicate a reduction in depressive-like symptoms post-sepsis and the psychoactive effects of the compound. Furthermore, a notable decrease in GFAP expression in the study highlights the compound's impact on mitigating sepsis-induced astrogliosis. This study demonstrates the effectiveness of 25H-NBOMe, a psychedelic in the phenethylamine class, in treating post-sepsis depression and reducing astrogliosis. However, the psychedelic nature of 25H-NBOMe calls for further investigation into similar compounds with less psychoactive impact, crucial for advancing treatment options for neuropsychiatric symptoms following sepsis.

Keywords: Animal models; Forced swimming test; Long-term sequelae; Neuroinflammation; Phenethylamine; Sepsis-associated encephalopathy.

MeSH terms

  • Animals
  • Depression* / drug therapy
  • Depression* / etiology
  • Hallucinogens / pharmacology
  • Hallucinogens / therapeutic use
  • Male
  • Phenethylamines / pharmacology
  • Phenethylamines / therapeutic use
  • Prefrontal Cortex / drug effects
  • Prefrontal Cortex / metabolism
  • Rats
  • Rats, Wistar*
  • Sepsis* / complications
  • Sepsis* / drug therapy
  • Sepsis* / metabolism
  • Sepsis* / psychology
  • Sepsis-Associated Encephalopathy / drug therapy
  • Sepsis-Associated Encephalopathy / metabolism

Substances

  • Hallucinogens
  • Phenethylamines