Anti-TL1A monoclonal antibody modulates the dysregulation of Th1/Th17 cells and attenuates granuloma formation in sarcoidosis by inhibiting the PI3K/AKT signaling pathway

Int Immunopharmacol. 2024 Aug 20:137:112360. doi: 10.1016/j.intimp.2024.112360. Epub 2024 Jun 8.

Abstract

Sarcoidosis is a systemic granulomatous disease characterized by non-caseating epithelioid cell granulomas. One of its immunological hallmarks is the differentiation of CD4 + naïve T cells into Th1/Th17 cells, accompanied by the release of numerous pro-inflammatory cytokines. The TL1A/DR3 signaling pathway plays a crucial role in activating effector lymphocytes, thereby triggering pro-inflammatory responses. The primary aim of this investigation was to scrutinize the impact of anti-TL1A monoclonal antibody on the dysregulation of Th1/Th17 cells and granuloma formation in sarcoidosis. Initially, the abnormal activation of the TL1A/DR3 signaling pathway in pulmonary tissues of sarcoidosis patients was confirmed using qPCR and immunohistochemistry techniques. Subsequently, employing a murine model of sarcoidosis, the inhibitory effects of anti-TL1A monoclonal antibody on the TL1A/DR3 signaling pathway in sarcoidosis were investigated through qPCR, immunohistochemistry, and Western blot experiments. The influence of anti-TL1A monoclonal antibody on granulomas was assessed through HE staining, while their effects on sarcoidosis Th1/Th17 cells and associated cytokine mRNA levels were evaluated using flow cytometry and qPCR, respectively. Immunofluorescence and Western blot experiments corroborated the inhibitory effects of anti-TL1A monoclonal antibody on the aberrant activation of the PI3K/AKT signaling pathway in sarcoidosis. The findings of this study indicate that the TL1A/DR3 signaling pathway is excessively activated in sarcoidosis. Anti-TL1A monoclonal antibody effectively inhibit this abnormal activation in sarcoidosis, thereby alleviating the dysregulation of Th1/Th17 cells and reducing the formation of pulmonary granulomas. This effect may be associated with the inhibition of the downstream PI3K/AKT signaling pathway. Anti-TL1A monoclonal antibody hold promise as a potential novel therapeutic intervention for sarcoidosis.

Keywords: Adaptive immunity; Anti-TL1A monoclonal antibody; Granuloma; Sarcoidosis.

MeSH terms

  • Adult
  • Animals
  • Antibodies, Monoclonal* / pharmacology
  • Antibodies, Monoclonal* / therapeutic use
  • Cytokines / immunology
  • Cytokines / metabolism
  • Disease Models, Animal
  • Female
  • Granuloma* / drug therapy
  • Granuloma* / immunology
  • Humans
  • Lung / immunology
  • Lung / pathology
  • Male
  • Mice
  • Mice, Inbred BALB C
  • Middle Aged
  • Phosphatidylinositol 3-Kinases* / immunology
  • Phosphatidylinositol 3-Kinases* / metabolism
  • Proto-Oncogene Proteins c-akt* / immunology
  • Proto-Oncogene Proteins c-akt* / metabolism
  • Receptors, Tumor Necrosis Factor, Member 25 / immunology
  • Receptors, Tumor Necrosis Factor, Member 25 / metabolism
  • Sarcoidosis* / drug therapy
  • Sarcoidosis* / immunology
  • Signal Transduction* / drug effects
  • Th1 Cells* / immunology
  • Th17 Cells* / immunology
  • Tumor Necrosis Factor Ligand Superfamily Member 15* / immunology
  • Tumor Necrosis Factor Ligand Superfamily Member 15* / metabolism

Substances

  • Antibodies, Monoclonal
  • Phosphatidylinositol 3-Kinases
  • Proto-Oncogene Proteins c-akt
  • Tumor Necrosis Factor Ligand Superfamily Member 15
  • Receptors, Tumor Necrosis Factor, Member 25
  • Tnfsf15 protein, mouse
  • Cytokines