Cytomegalovirus Antiviral Resistance Among Kidney Transplant Recipients in a Phase 3 Trial of Letermovir vs Valganciclovir Prophylaxis

J Infect Dis. 2024 Dec 16;230(6):e1287-e1298. doi: 10.1093/infdis/jiae287.

Abstract

Background: In a phase 3 trial, letermovir was noninferior to valganciclovir for cytomegalovirus (CMV) disease prophylaxis in kidney transplant recipients who were CMV-seronegative and received kidneys from donors who were CMV-seropositive. Genotypic antiviral resistance and CMV glycoprotein B (gB) genotype are reported.

Methods: Plasma samples with detectable CMV DNA were sequenced for the presence of known letermovir and valganciclovir resistance-associated amino acid substitutions (RASs) encoded by CMV gene regions (UL51, UL54, UL56, UL89, UL97) and prevalence of gB (UL55) genotypes (gB1-gB5).

Results: Among participants, 84 of 292 (letermovir) and 93 of 297 (valganciclovir) had evaluable data for ≥1 gene target. Letermovir RASs were not detected in participants who received letermovir prophylaxis; however, 3 had valganciclovir RASs (pUL97). Twelve participants who received valganciclovir prophylaxis had valganciclovir RASs (pUL54, pUL97), and 1 who did not receive letermovir during the trial had letermovir RASs (pUL56). All but 1 participant responded to valganciclovir treatment irrespective of breakthrough CMV DNAemia or frequency of RASs. gB1 was the most frequent genotype across all participants and subgroups.

Conclusions: Letermovir RASs were not detected with letermovir prophylaxis, supporting a low risk for development of resistance in kidney transplant recipients who were CMV-seronegative and received kidneys from donors who were CMV-seropositive.

Clinical trials registration: ClinicalTrials.gov, NCT03443869; EudraCT, 2017-001055-30.

Keywords: cytomegalovirus; kidney transplant recipient; letermovir; prophylaxis; resistance.

Publication types

  • Clinical Trial, Phase III
  • Randomized Controlled Trial

MeSH terms

  • Acetates / pharmacology
  • Acetates / therapeutic use
  • Adult
  • Antiviral Agents* / therapeutic use
  • Cytomegalovirus Infections* / epidemiology
  • Cytomegalovirus Infections* / prevention & control
  • Cytomegalovirus Infections* / virology
  • Cytomegalovirus* / drug effects
  • Cytomegalovirus* / genetics
  • Drug Resistance, Viral* / genetics
  • Female
  • Ganciclovir / analogs & derivatives
  • Ganciclovir / therapeutic use
  • Genotype*
  • Humans
  • Kidney Transplantation*
  • Male
  • Middle Aged
  • Quinazolines* / therapeutic use
  • Transplant Recipients*
  • Valganciclovir* / therapeutic use

Substances

  • Antiviral Agents
  • Valganciclovir
  • letermovir
  • Quinazolines
  • Acetates
  • Ganciclovir

Associated data

  • ClinicalTrials.gov/NCT03443869