A phase 1 study of biweekly nab-paclitaxel/oxaliplatin/S-1/LV for advanced upper gastrointestinal cancers: TCOG T1216 study

Oncologist. 2024 Oct 3;29(10):e1396-e1405. doi: 10.1093/oncolo/oyae109.

Abstract

Background: Oxaliplatin- and fluoropyrimidine-based triplet regimens have demonstrated feasibility and efficacy in the treatment of upper gastrointestinal (UGI) cancers. Herein, we evaluate the feasibility and preliminary efficacy of biweekly nab-paclitaxel plus oxaliplatin and S-1/leucovorin (SOLAR) in chemonaïve UGI cancers.

Methods: A 3 + 3 phase 1 study was conducted to determine the maximal tolerated dose (MTD) of oxaliplatin in SOLAR (nab-paclitaxel [150 mg/m2 in D1], oxaliplatin [60, 75, or 85 mg/m2 in D1], and oral S-1/leucovorin [35 mg/m2 and 30 mg bid from D1 to D7]). The secondary endpoints were overall response rate (ORR), progression-free survival (PFS), overall survival (OS), and safety.

Results: Thirteen and 6 accruals were in the dose-escalation and MTD expansion cohorts, respectively. One of 6 patients at level III experienced dose-limiting toxicity (grade 3 diarrhea), which revealed that the MTD of oxaliplatin was 85 mg/m2. After a mean of 15.9 cycles of treatment, the most common treatment-related grade 3/4 toxicities were neutropenia (57.9%) and diarrhea (21.1%). The ORR was 63.2%. The median PFS and OS were 12.5 and 24.7 months, respectively.

Conclusion: The current study revealed the MTD of oxaliplatin and demonstrated the preliminary efficacy of SOLAR in UGI cancers, which deserves further investigation.

Clinicaltrials.gov identifier: NCT03162510.

Keywords: S-1/leucovorin; nab-paclitaxel; oxaliplatin; phase 1; upper gastrointestinal cancers.

Publication types

  • Clinical Trial, Phase I
  • Multicenter Study

MeSH terms

  • Adult
  • Aged
  • Albumins* / administration & dosage
  • Albumins* / adverse effects
  • Albumins* / pharmacology
  • Albumins* / therapeutic use
  • Antineoplastic Combined Chemotherapy Protocols* / adverse effects
  • Antineoplastic Combined Chemotherapy Protocols* / pharmacology
  • Antineoplastic Combined Chemotherapy Protocols* / therapeutic use
  • Drug Combinations*
  • Female
  • Gastrointestinal Neoplasms* / drug therapy
  • Gastrointestinal Neoplasms* / mortality
  • Gastrointestinal Neoplasms* / pathology
  • Humans
  • Leucovorin* / administration & dosage
  • Leucovorin* / therapeutic use
  • Male
  • Maximum Tolerated Dose
  • Middle Aged
  • Oxaliplatin* / administration & dosage
  • Oxaliplatin* / pharmacology
  • Oxaliplatin* / therapeutic use
  • Oxonic Acid* / administration & dosage
  • Oxonic Acid* / adverse effects
  • Oxonic Acid* / therapeutic use
  • Paclitaxel* / administration & dosage
  • Paclitaxel* / adverse effects
  • Paclitaxel* / pharmacology
  • Paclitaxel* / therapeutic use
  • Tegafur* / administration & dosage
  • Tegafur* / adverse effects
  • Tegafur* / therapeutic use

Substances

  • Oxaliplatin
  • Paclitaxel
  • 130-nm albumin-bound paclitaxel
  • Drug Combinations
  • Oxonic Acid
  • S 1 (combination)
  • Albumins
  • Leucovorin
  • Tegafur

Associated data

  • ClinicalTrials.gov/NCT03162510