TXNDC5 Plays a Crucial Role in Regulating Endoplasmic Reticulum Activity through Different ER Stress Signaling Pathways in Hepatic Cells

Int J Mol Sci. 2024 Jun 28;25(13):7128. doi: 10.3390/ijms25137128.

Abstract

The pathogenesis of non-alcoholic fatty liver disease (NAFLD) is influenced by a number of variables, including endoplasmic reticulum stress (ER). Thioredoxin domain-containing 5 (TXNDC5) is a member of the protein disulfide isomerase family and acts as an endoplasmic reticulum (ER) chaperone. Nevertheless, the function of TXNDC5 in hepatocytes under ER stress remains largely uncharacterized. In order to identify the role of TXNDC5 in hepatic wild-type (WT) and TXNDC5-deficient (KO) AML12 cell lines, tunicamycin, palmitic acid, and thapsigargin were employed as stressors. Cell viability, mRNA, protein levels, and mRNA splicing were then assayed. The protein expression results of prominent ER stress markers indicated that the ERN1 and EIF2AK3 proteins were downregulated, while the HSPA5 protein was upregulated. Furthermore, the ATF6 protein demonstrated no significant alterations in the absence of TXNDC5 at the protein level. The knockout of TXNDC5 has been demonstrated to increase cellular ROS production and its activity is required to maintain normal mitochondrial function during tunicamycin-induced ER stress. Tunicamycin has been observed to disrupt the protein levels of HSPA5, ERN1, and EIF2AK3 in TXNDC5-deficient cells. However, palmitic acid has been observed to disrupt the protein levels of ATF6, HSPA5, and EIF2AK3. In conclusion, TXNDC5 can selectively activate distinct ER stress pathways via HSPA5, contingent on the origin of ER stress. Conversely, the absence of TXNDC5 can disrupt the EIF2AK3 cascade.

Keywords: ATF6; EIF2AK3; ERN1; HSPA5; IRE1a; NAFLD; PERK; TXNDC5; endoplasmic reticulum stress; hepatocytes; liver; palmitic acid; thapsigargin; tunicamycin.

MeSH terms

  • Activating Transcription Factor 6 / genetics
  • Activating Transcription Factor 6 / metabolism
  • Animals
  • Cell Line
  • Cell Survival / drug effects
  • Endoplasmic Reticulum Chaperone BiP* / metabolism
  • Endoplasmic Reticulum Stress*
  • Endoplasmic Reticulum* / metabolism
  • Endoribonucleases / genetics
  • Endoribonucleases / metabolism
  • Heat-Shock Proteins / genetics
  • Heat-Shock Proteins / metabolism
  • Hepatocytes* / metabolism
  • Humans
  • Mice
  • Non-alcoholic Fatty Liver Disease / genetics
  • Non-alcoholic Fatty Liver Disease / metabolism
  • Non-alcoholic Fatty Liver Disease / pathology
  • Palmitic Acid / metabolism
  • Palmitic Acid / pharmacology
  • Protein Disulfide-Isomerases* / genetics
  • Protein Disulfide-Isomerases* / metabolism
  • Protein Serine-Threonine Kinases / genetics
  • Protein Serine-Threonine Kinases / metabolism
  • Reactive Oxygen Species / metabolism
  • Signal Transduction*
  • Thapsigargin / pharmacology
  • Thioredoxins / genetics
  • Thioredoxins / metabolism
  • Tunicamycin* / pharmacology

Substances

  • Endoplasmic Reticulum Chaperone BiP
  • Protein Disulfide-Isomerases
  • Tunicamycin
  • Hspa5 protein, mouse
  • Reactive Oxygen Species
  • Activating Transcription Factor 6
  • Protein Serine-Threonine Kinases
  • HSPA5 protein, human
  • Heat-Shock Proteins
  • Endoribonucleases
  • Palmitic Acid
  • Thapsigargin
  • PC-TRP protein, mouse
  • Thioredoxins
  • Atf6 protein, mouse