Anti-tuberculosis effect of microbiome therapeutic PMC205 in extensively drug-resistant pulmonary tuberculosis in vivo

Int J Antimicrob Agents. 2024 Sep;64(3):107274. doi: 10.1016/j.ijantimicag.2024.107274. Epub 2024 Jul 11.

Abstract

Background: Tuberculosis is a highly contagious disease caused by Mycobacterium tuberculosis, and the increase in antibiotic resistance threatens humankind. Therefore, there is an urgent need to develop new anti-tuberculosis drugs that can overcome the limitations of existing drugs. Here, we report the anti-tuberculosis effect of microbiome therapeutic PMC205, a strain of Bacillus subtilis.

Methods: The anti-tuberculosis activity of probiotics was evaluated in mouse models of lethal and latent pulmonary tuberculosis induced by high or low-dose infection of the extensively drug-resistant strain. Probiotics were administered by inhalation, and the burden of M. tuberculosis in the lungs, along with mortality and clinical observations, were monitored for 12 weeks and 8 months, respectively. For an in-depth understanding, analysis of the microbiome and inflammatory profile of the lung microenvironment and induction of autophagy in vitro were explored.

Results: After inhalation administration of PMC205 for 3 months, the survival rate was 100%, unlike all deaths in the saline-treated group, and the burden of M. tuberculosis in the lungs was reduced by log 1.3 in the 8-month latent tuberculosis model. Moreover, PMC205 induced recovery of disrupted lung microflora, increased butyric acid, and suppressed excessive inflammation. It also promoted autophagy.

Conclusions: These results confirm PMC205's anti-tuberculosis effect, suggesting that it can be developed as an adjuvant to current antibiotic therapy to solve the drug-resistant tuberculosis problem.

Keywords: Adjuvant microbiome therapeutic; Autophagy; Mycobacterium tuberculosis; Tuberculosis; XDR (extensively drug-resistant).

MeSH terms

  • Animals
  • Antitubercular Agents* / pharmacology
  • Antitubercular Agents* / therapeutic use
  • Autophagy / drug effects
  • Bacillus subtilis / drug effects
  • Disease Models, Animal*
  • Extensively Drug-Resistant Tuberculosis* / drug therapy
  • Extensively Drug-Resistant Tuberculosis* / microbiology
  • Female
  • Humans
  • Lung* / microbiology
  • Lung* / pathology
  • Mice
  • Mice, Inbred C57BL
  • Microbiota* / drug effects
  • Mycobacterium tuberculosis* / drug effects
  • Probiotics* / administration & dosage
  • Probiotics* / therapeutic use
  • Tuberculosis, Pulmonary* / drug therapy
  • Tuberculosis, Pulmonary* / microbiology

Substances

  • Antitubercular Agents