Myocarditis Following Pembrolizumab Plus Axitinib, and Belzutifan Plus Lenvatinib for Renal Cell Carcinoma: A Case Report

Cardiovasc Toxicol. 2024 Nov;24(11):1168-1173. doi: 10.1007/s12012-024-09906-w. Epub 2024 Jul 31.

Abstract

Cardiac toxicity is an adverse event of several classes of anti-cancer drugs. Herein, we present the case of a 52-year-old woman with metastatic renal cell carcinoma (RCC), previously treated with debulking surgery, pembrolizumab (immune checkpoint inhibitor) in combination with axitinib (tyrosine kinase inhibitor (TKI)), followed by lenvatinib (TKI) and belzutifan (HIF-2α inhibitor), who developed myocarditis proven by cardiac magnetic resonance and endomyocardial biopsy. The case was notable for reporting a not-yet described adverse event during treatment with belzutifan plus lenvatinib, the etiology of which was of unobvious determination given the pre-exposure to pembrolizumab, a known cause of drug-related myocarditis. We surmise that myocarditis was a delayed adverse event related to pembrolizumab (8 months after treatment interruption), although we emphasize that only attentive monitoring of cardiac adverse events of patients exposed to belzutifan and lenvatinib in the context of large clinical trials may rule out any causal implication of these drugs.

Keywords: Chemotherapy; Immune checkpoint inhibitors; Immunotherapy; Myocarditis; Renal cell carcinoma.

Publication types

  • Case Reports

MeSH terms

  • Antibodies, Monoclonal, Humanized* / adverse effects
  • Antineoplastic Combined Chemotherapy Protocols* / adverse effects
  • Axitinib* / adverse effects
  • Carcinoma, Renal Cell* / drug therapy
  • Female
  • Humans
  • Immune Checkpoint Inhibitors / adverse effects
  • Kidney Neoplasms* / drug therapy
  • Kidney Neoplasms* / pathology
  • Middle Aged
  • Myocarditis* / chemically induced
  • Myocarditis* / diagnosis
  • Phenylurea Compounds* / adverse effects
  • Protein Kinase Inhibitors / adverse effects
  • Quinolines* / adverse effects
  • Treatment Outcome

Substances

  • lenvatinib
  • Quinolines
  • pembrolizumab
  • Antibodies, Monoclonal, Humanized
  • Axitinib
  • Phenylurea Compounds
  • Protein Kinase Inhibitors
  • Immune Checkpoint Inhibitors