Metabolism of 4,7,10,13,16-docosapentaenoic acid by human platelet cyclooxygenase and lipoxygenase

Biochim Biophys Acta. 1985 Jun 14;835(1):29-35. doi: 10.1016/0005-2760(85)90026-8.

Abstract

Washed human platelets are shown to metabolize 4,7,10,13,16-docosapentaenoic acid into three major metabolites which were purified by reverse-phase HPLC. The mass spectra of the methyl ester-trimethylsilyl ether and ethyl ester-trimethylsilyl ether of compound A established it as delta 4-dihomo-thromboxane B2. Compound B was shown to be 14-hydroxy-4,7,10,12-nonadecatetraenoic acid, which is analogous to 12-hydroxy-5,8,10-heptadecatrienoic acid from arachidonic acid. Compound C was produced via an indomethacin-insensitive pathway and was identified as 14-hydroxy-4,7,10,12,16-docosapentaenoic acid. Time- and substrate-dependent studies showed that compounds A,B and C were produced approximately 10,15 and 65% of the extent to which thromboxane B2, 12-hydroxy-5,8,10-heptadecatrienoic acid and 12-hydroxy-5,8,10,14-eicosatetraenoic acid were produced, respectively, from arachidonic acid.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Arachidonic Acid
  • Arachidonic Acids / blood
  • Blood Platelets / enzymology*
  • Chromatography, High Pressure Liquid
  • Chromatography, Thin Layer
  • Fatty Acids, Unsaturated / blood*
  • Humans
  • Lipoxygenase / blood*
  • Mass Spectrometry
  • Prostaglandin-Endoperoxide Synthases / blood*
  • Time Factors

Substances

  • Arachidonic Acids
  • Fatty Acids, Unsaturated
  • Arachidonic Acid
  • Lipoxygenase
  • Prostaglandin-Endoperoxide Synthases
  • docosapentaenoic acid