Ultra-low dose estradiol and dydrogesterone for the treatment of menopausal symptoms in a pooled, multi-ethnic population

Maturitas. 2024 Dec:190:108117. doi: 10.1016/j.maturitas.2024.108117. Epub 2024 Sep 17.

Abstract

Objectives: Evidence suggests ethnicity-specific differences in postmenopausal symptoms, highlighting the need for therapies that are efficacious across different ethnicities. We evaluated the efficacy of an ultra-low dose combination of 0.5 mg estradiol and 0.25 mg dydrogesterone (E 0.5 mg/D 2.5 mg) in alleviating vasomotor symptoms across a multi-ethnic population.

Study design: Data from two controlled trials were pooled to form a dataset of 583 postmenopausal women from across Europe and China. Participants were randomized to receive treatment with E 0.5 mg/D 2.5 mg or placebo for 12 weeks.

Main outcome measures: The main efficacy variable was absolute change in the number of hot flushes from baseline to end of treatment. Health-related quality of life and safety were also assessed.

Results: Change in the number of hot flushes per day was greater with E 0.5 mg/D 2.5 mg versus placebo (mean difference - 1.5, 95 % confidence interval - 2.1, -1.0; p < 0.001). Participants treated with E 0.5 mg/D 2.5 mg reported improvement in health-related quality of life (including psychological symptoms, vaginal dryness), and high amenorrhea rates. Combined E 0.5 mg/D 2.5 mg was well tolerated: there were no differences between groups in the percentage of participants with at least one serious adverse event or treatment-emergent serious adverse events. Analysis of change in body weight indicated no differences between groups.

Conclusions: This pooled analysis demonstrates the consistent efficacy of E 0.5 mg/D 2.5 mg in the treatment of menopause-related symptoms across a multi-ethnic population of postmenopausal women.

Keywords: Dydrogesterone; Estradiol; Menopause hormone therapy; Ultra-low dose; Vasomotor symptoms.

Publication types

  • Randomized Controlled Trial

MeSH terms

  • Aged
  • China / ethnology
  • Dydrogesterone* / administration & dosage
  • Dydrogesterone* / therapeutic use
  • Estradiol* / administration & dosage
  • Estrogen Replacement Therapy / methods
  • Ethnicity
  • Europe
  • Female
  • Hot Flashes* / drug therapy
  • Hot Flashes* / ethnology
  • Humans
  • Menopause / drug effects
  • Menopause / ethnology
  • Middle Aged
  • Postmenopause
  • Progestins / administration & dosage
  • Progestins / therapeutic use
  • Quality of Life*

Substances

  • Dydrogesterone
  • Estradiol
  • Progestins