Pharmacologic or genetic targeting of peripheral nerves prevents peri-articular traumatic heterotopic ossification

Bone Res. 2024 Sep 26;12(1):54. doi: 10.1038/s41413-024-00358-0.

Abstract

Heterotopic ossification (HO) is a pathological process that commonly arises following severe polytrauma, characterized by the anomalous differentiation of mesenchymal progenitor cells and resulting in the formation of ectopic bone in non-skeletal tissues. This abnormal bone growth contributes to pain and reduced mobility, especially when adjacent to a joint. Our prior observations suggested an essential role of NGF (Nerve Growth Factor)-responsive TrkA (Tropomyosin Receptor Kinase A)-expressing peripheral nerves in regulating abnormal osteochondral differentiation following tendon injury. Here, we utilized a recently developed mouse model of hip arthroplasty-induced HO to further validate the role of peripheral nerve regulation of traumatic HO. Nerve ingrowth was either modulated using a knockin transgenic animals with point mutation in TrkA, or local treatment with an FDA-approved formulation of long acting Bupivacaine which prevents peripheral nerve growth. Results demonstrate exuberant sensory and sympathetic nerve growth within the peri-articular HO site, and that both methods to reduce local innervation significantly reduced heterotopic bone formation. TrkA inhibition led to a 34% reduction in bone volume, while bupivacaine treatment resulted in a 50% decrease. Mechanistically, alterations in TGFβ and FGF signaling activation accompanied both methods of local denervation, and a shift in macrophages from M1 to M2 phenotypes was observed. In sum, these studies reinforce the observations that peripheral nerves play a role in the etiopathogenesis of HO, and that targeting local nerves represents a potential therapeutic approach for disease prevention.

MeSH terms

  • Animals
  • Bupivacaine* / administration & dosage
  • Bupivacaine* / pharmacology
  • Mice
  • Mice, Inbred C57BL
  • Mice, Transgenic
  • Ossification, Heterotopic* / genetics
  • Ossification, Heterotopic* / pathology
  • Ossification, Heterotopic* / prevention & control
  • Peripheral Nerves* / drug effects
  • Peripheral Nerves* / metabolism
  • Peripheral Nerves* / pathology
  • Receptor, trkA* / genetics
  • Receptor, trkA* / metabolism
  • Transforming Growth Factor beta / genetics
  • Transforming Growth Factor beta / metabolism

Substances

  • Bupivacaine
  • Receptor, trkA
  • Transforming Growth Factor beta