Effects of tenofovir alafenamide fumarate on serum lipid profiles in patients with chronic hepatitis B

Virol J. 2024 Sep 28;21(1):234. doi: 10.1186/s12985-024-02515-7.

Abstract

Background: Concerns have been raised regarding changes in lipid profiles among patients with chronic hepatitis B (CHB) during tenofovir alafenamide fumarate (TAF) treatment. We aimed to evaluate the effect of TAF treatment on the lipid profiles of patients with CHB.

Methods: A total of 430 patients with CHB from three hospitals were retrospectively included, including 158 patients treated with TAF and 272 patients treated with tenofovir disoproxil fumarate (TDF).

Results: In this multicenter cohort, the cumulative incidence of dyslipidemia was notably higher in the TAF group than in the TDF group (P < 0.001). After TAF treatment, a significant elevation was observed in triglyceride (TG) levels (from 0.83 mmol/L to 1.02 mmol/L, P < 0.001) and total cholesterol (TC) levels (from 4.16 mmol/L to 4.32 mmol/L, P < 0.001). Similar changes in TG and TC levels were observed in the TAF group after propensity score matching (PSM). The TG levels (from 0.83 mmol/L to 1.04 mmol/L, P < 0.001) and TC levels (from 4.16 mmol/L to 4.38 mmol/L, P < 0.001) were both increased significantly compared to the baseline levels in the PSM cohort of patients treated with TAF. TAF treatment was independently associated with elevated TG levels (HR = 2.800, 95% CI: 1.334-5.876, P = 0.006) and TC levels (HR = 9.045, 95% CI: 3.836-21.328, P < 0.001).

Conclusions: Compared with TDF treatment, TAF treatment was associated with dyslipidemia in patients with CHB. Close monitoring of lipid profiles is needed in patients with CHB who received TAF treatment.

Keywords: Chronic hepatitis B; Tenofovir alafenamide fumarate; Total cholesterol; Triglyceride.

Publication types

  • Multicenter Study

MeSH terms

  • Adenine / analogs & derivatives
  • Adenine / therapeutic use
  • Adult
  • Alanine* / therapeutic use
  • Antiviral Agents* / therapeutic use
  • Cholesterol / blood
  • Dyslipidemias / blood
  • Dyslipidemias / chemically induced
  • Dyslipidemias / drug therapy
  • Female
  • Hepatitis B, Chronic* / blood
  • Hepatitis B, Chronic* / drug therapy
  • Hepatitis B, Chronic* / virology
  • Humans
  • Lipids* / blood
  • Male
  • Middle Aged
  • Retrospective Studies
  • Tenofovir* / analogs & derivatives
  • Tenofovir* / therapeutic use
  • Triglycerides / blood

Substances

  • Tenofovir
  • tenofovir alafenamide
  • Antiviral Agents
  • Alanine
  • Lipids
  • Adenine
  • Triglycerides
  • Cholesterol