Long-term safety and efficacy of ropeginterferon alfa-2b in Japanese patients with polycythemia vera

Int J Hematol. 2024 Dec;120(6):675-683. doi: 10.1007/s12185-024-03846-5. Epub 2024 Oct 3.

Abstract

Ropeginterferon alfa-2b (ropegIFN), a new-generation interferon-based agent, has been approved in Japan for patients with polycythemia vera (PV) who are ineligible for or respond inadequately to conventional treatment. However, long-term outcomes with ropegIFN in Japanese patients have not been reported. This extension of a phase 2 study of ropegIFN in Japanese patients with PV aimed to determine its long-term safety/efficacy, and changes over time in JAK2 V617F allele burden. Here, we report data from the phase 2 study and subsequent extension over a period of 36 months. The primary endpoint was the complete hematologic response (CHR) maintenance rate without phlebotomy (hematocrit value < 45% without phlebotomy during the previous 12 weeks, platelet count ≤ 400 × 109/L, and white blood cell count ≤ 10 × 109/L). The CHR maintenance rates were 8/27 (29.6%), 18/27 (66.7%), and 22/27 (81.5%) at 12, 24, and 36 months, respectively. No thrombotic or hemorrhagic events occurred. The median allele burden change from baseline was - 74.8% at 36 months. All patients experienced adverse events; 25/27 (92.6%) experienced adverse drug reactions (ADRs), but no serious ADRs or deaths occurred. This interim analysis demonstrated the safety and efficacy of ropegIFN over 36 months in Japanese patients with PV.

Keywords: JAK2 V617F allele burden; Hematologic response; Molecular response; Polycythemia vera; Ropeginterferon alfa-2b.

Publication types

  • Clinical Trial, Phase II
  • Multicenter Study

MeSH terms

  • Adult
  • Aged
  • Aged, 80 and over
  • Alleles
  • East Asian People
  • Female
  • Humans
  • Interferon alpha-2* / administration & dosage
  • Interferon alpha-2* / adverse effects
  • Interferon alpha-2* / therapeutic use
  • Interferon-alpha* / administration & dosage
  • Interferon-alpha* / adverse effects
  • Interferon-alpha* / therapeutic use
  • Janus Kinase 2* / genetics
  • Japan
  • Male
  • Middle Aged
  • Polycythemia Vera* / drug therapy
  • Polycythemia Vera* / genetics
  • Polyethylene Glycols* / administration & dosage
  • Polyethylene Glycols* / adverse effects
  • Polyethylene Glycols* / therapeutic use
  • Recombinant Proteins* / administration & dosage
  • Recombinant Proteins* / adverse effects
  • Recombinant Proteins* / therapeutic use
  • Time Factors
  • Treatment Outcome

Substances

  • Interferon alpha-2
  • Interferon-alpha
  • JAK2 protein, human
  • Janus Kinase 2
  • peginterferon alfa-2b
  • Polyethylene Glycols
  • Recombinant Proteins