Dose sparing enabled by immunization with influenza vaccine using orally dissolving film

Int J Pharm. 2024 Dec 25;667(Pt B):124945. doi: 10.1016/j.ijpharm.2024.124945. Epub 2024 Nov 15.

Abstract

Influenza vaccine delivered by orally dissolving film vaccine (ODFV) is a promising approach. In this study, we generated three ODFVs each comprising pulluan and trehalose with different doses of inactivated A/Puerto Rico/8/34, H1N1 virus (ODFV I, II, III) to evaluate their dose-sparing effect in mice. The ODFVs were placed on the tongues of mice to elicit immunization and after 3 immunizations at 4-week intervals, mice were challenged with a lethal dose of A/PR/8/34 to assess vaccine-induced protection. The 3 ODFVs containing 50, 250, or 750 μg of inactivated viruses elicited virus-specific antibody responses and virus neutralization in a dose-dependent manner. Dose-dependent antibody responses were also observed from the mucosal tissue samples, and also from antibody-secreting cells of the lungs and spleens. ODFV-induced cellular immunity, particularly germinal center B cells and T cells were also dose-dependent. Importantly, all 3 ODFVs evaluated in this study provided complete protection by strongly suppressing the pro-inflammatory cytokine production and lung virus titers. None of the immunized mice underwent noticeable weight loss nor succumbed to death, a phenomenon that was only observed in the infection challenge controls. These results indicated that the protection conferred by a low dose influenza vaccine formulated in ODF is comparable to that of a high-dose vaccine, thereby enabling vaccine dose sparing effect.

Keywords: Dose-sparing effect; Influenza virus; Orally dissolving film; Vaccination.

MeSH terms

  • Administration, Oral
  • Animals
  • Antibodies, Viral / blood
  • Cytokines
  • Dose-Response Relationship, Immunologic
  • Female
  • Immunization / methods
  • Influenza A Virus, H1N1 Subtype* / immunology
  • Influenza Vaccines* / administration & dosage
  • Influenza Vaccines* / immunology
  • Lung / immunology
  • Lung / virology
  • Mice
  • Mice, Inbred BALB C*
  • Orthomyxoviridae Infections* / immunology
  • Orthomyxoviridae Infections* / prevention & control
  • Trehalose / administration & dosage
  • Vaccines, Inactivated / administration & dosage
  • Vaccines, Inactivated / immunology

Substances

  • Influenza Vaccines
  • Antibodies, Viral
  • Trehalose
  • Vaccines, Inactivated
  • Cytokines