Mechanochemically facilitated silver-catalyzed direct H/D exchange on heteroarenes

Org Biomol Chem. 2025 Jan 2;23(2):297-302. doi: 10.1039/d4ob01581a.

Abstract

Despite recent advances in H/D exchange, the effective deuteration of polyarenes remains challenging, due to their insolubility and hydrophobicity. This study presents a concept proofing of a mechanochemically facilitated direct H/D exchange. The silver-catalyzed deuteration of heteroarenes was promoted smoothly within 99 minutes of grinding, with heavy water as the deuterium source.