Bicyclic compounds with potential antiulcer and/or antisecretory activity. II. 1(or 3),4,6,7-Tetrahydro-1(3)H-pyrano[3,4-d]imidazoles and 1(or 3),4,6,7-tetrahydro-1(3)H-thiopyrano[3,4-d]imidazoles

Farmaco Sci. 1986 Jan;41(1):23-40.

Abstract

Owing to our current interest in synthesizing and evaluating the antiulcer and antisecretory activity of bicyclic compounds, a series of 1(or 3),4,6,7-tetrahydropyrano- and 1(or 3),4,6,7-tetrahydrothiopyrano-[3,4-d]imidazoles was synthesized and tested. The biological results were compared with those of some previously described 4,5,6,7-tetrahydroimidazo-[4,5-c]pyridine and 4,5,6,7-tetrahydrobenzimidazole derivatives.

MeSH terms

  • Animals
  • Anti-Ulcer Agents / chemical synthesis*
  • Chemical Phenomena
  • Chemistry
  • Chemistry, Physical
  • Gastric Juice / metabolism
  • Guinea Pigs
  • Imidazoles / chemical synthesis*
  • Imidazoles / pharmacology
  • Mice
  • Pyrans / chemical synthesis*
  • Pyrans / pharmacology
  • Rats
  • Stomach Ulcer / etiology
  • Stomach Ulcer / physiopathology
  • Stomach Ulcer / prevention & control*
  • Stress, Psychological / complications

Substances

  • Anti-Ulcer Agents
  • Imidazoles
  • Pyrans