Olmesartan: 360-degree Perspectives Befitting an Angiotensin Receptor Blocker

J Assoc Physicians India. 2024 Dec;72(12):59-72. doi: 10.59556/japi.72.0780.

Abstract

India has a high burden of hypertension (HTN), which is often poorly controlled, leading to hypertension-mediated organ damage (HMOD). In the management of HTN, angiotensin receptor blockers (ARBs) assume prime importance, being first-line agents for most patient subgroups. Olmesartan is a highly efficacious ARB that demonstrates sustained blood pressure (BP) reduction over 24 hours. Moreover, it also assumes a protective role by reducing microvascular inflammation, left ventricular hypertrophy, proteinuria, vascular stiffness, central aortic BP, cardiocerebrovascular events and atrial fibrillation. To enhance therapeutic compliance and achieve BP goals, single-pill combinations with other antihypertensive agents are also available. This review holistically summarizes the evidence of olmesartan for HTN management for not only BP reduction but also organoprotective effects.

Publication types

  • Review

MeSH terms

  • Angiotensin II Type 1 Receptor Blockers* / therapeutic use
  • Antihypertensive Agents / therapeutic use
  • Blood Pressure / drug effects
  • Humans
  • Hypertension* / drug therapy
  • Imidazoles* / therapeutic use
  • Tetrazoles* / therapeutic use

Substances

  • olmesartan
  • Tetrazoles
  • Imidazoles
  • Angiotensin II Type 1 Receptor Blockers
  • Antihypertensive Agents