Defective glycosylation and ELFN1 binding of mGluR6 congenital stationary night blindness mutants

Life Sci Alliance. 2024 Dec 16;8(3):e202403118. doi: 10.26508/lsa.202403118. Print 2025 Mar.

Abstract

Synaptic transmission from photoreceptors to ON-bipolar cells (BCs) requires the postsynaptic metabotropic glutamate receptor mGluR6, located at BC dendritic tips. Binding of the neurotransmitter glutamate initiates G protein signaling that regulates the TRPM1 transduction channel. mGluR6 also interacts with presynaptic ELFN adhesion proteins, and these interactions are important for mGluR6 synaptic localization. The mechanisms of mGluR6 trafficking and synaptic targeting remain poorly understood. In this study, we investigated mGluR6 missense mutations from patients with congenital stationary night blindness (CSNB), which is associated with loss of synaptic transmission to ON-BCs. We found that multiple CSNB mutations in the extracellular ligand-binding domain of mGluR6 impart a trafficking defect leading to lack of complex N-glycosylation but efficient plasma membrane insertion, suggesting a Golgi bypass mechanism. These mutants fail to bind ELFN1, consistent with lack of a necessary modification normally acquired in the Golgi. The same mutants were mislocalized in bipolar cells, explaining the loss of function in CSNB. The results reveal a key role of Golgi trafficking in mGluR6 function, and suggest a role of the extracellular domain in Golgi sorting.

MeSH terms

  • Animals
  • Cell Membrane / metabolism
  • Congenital Disorders of Glycosylation / genetics
  • Congenital Disorders of Glycosylation / metabolism
  • Eye Diseases, Hereditary* / genetics
  • Eye Diseases, Hereditary* / metabolism
  • Genetic Diseases, X-Linked* / genetics
  • Genetic Diseases, X-Linked* / metabolism
  • Glycosylation
  • Golgi Apparatus* / metabolism
  • HEK293 Cells
  • Humans
  • Mutation
  • Mutation, Missense
  • Myopia* / genetics
  • Myopia* / metabolism
  • Night Blindness* / genetics
  • Night Blindness* / metabolism
  • Protein Binding
  • Protein Transport
  • Receptors, Glutamate
  • Receptors, Metabotropic Glutamate* / genetics
  • Receptors, Metabotropic Glutamate* / metabolism
  • Retinal Bipolar Cells / metabolism
  • Synaptic Transmission / genetics
  • TRPM Cation Channels / genetics
  • TRPM Cation Channels / metabolism

Substances

  • Receptors, Metabotropic Glutamate
  • metabotropic glutamate receptor 6
  • GRM6 protein, human
  • TRPM Cation Channels
  • Receptors, Glutamate

Supplementary concepts

  • Night blindness, congenital stationary

Associated data

  • PDB/7E9H
  • PDB/7EPC