Potential Contribution of Epithelial Growth Factor Receptor to PI3K/AKT Pathway Dysregulation in Canine Soft Tissue Sarcoma

In Vivo. 2025 Jan-Feb;39(1):110-119. doi: 10.21873/invivo.13808.

Abstract

Background/aim: Soft tissue sarcoma (STS) is a mesenchymal tumor affecting multiple organs in dogs. Previous studies identified activation of the phosphatidylinositol-3 kinase (PI3K)/protein kinase B (PKB, AKT) pathway in canine STS cell lines and clinical samples, but the underlying mechanism remains unclear. This study investigated PTEN loss, PIK3CA mutation, and EGFR over-expression as potential drivers of PI3K/AKT pathway activation in STS.

Materials and methods: We analyzed 36 canine STS samples. PTEN and EGFR expression were evaluated using immunohistochemistry, while PIK3CA and EGFR mutations were assessed through DNA sequencing.

Results: PTEN was expressed in all analyzed samples, with no evidence of loss. Weak PTEN expression was observed in 12 (33.3%) samples, while 24 (66.7%) showed normal expression. DNA sequencing of PIK3CA revealed a single point mutation (c.554 A>C, H554P) in one case, but no hotspot mutations were identified. High EGFR expression was significantly correlated with elevated phospho-AKT levels (p<0.0001). Immunolabelling indicated that 30 samples (83.3%) were EGFR-positive, and 27 of these also showed positive phospho-AKT labeling. Accordingly, one missense point mutation in exon 21 of EGFR (E868K) was identified in one of 12 samples.

Conclusion: EGFR over-expression, rather than PTEN loss or PIK3CA mutations, may contribute to PI3K/AKT pathway dysregulation in canine STS. Further studies with larger sample sizes and additional validation techniques are necessary to confirm these findings.

Keywords: Canine; EGFR; PIK3CA; PTEN; soft tissue sarcoma.

MeSH terms

  • Animals
  • Class I Phosphatidylinositol 3-Kinases / genetics
  • Class I Phosphatidylinositol 3-Kinases / metabolism
  • Dog Diseases / genetics
  • Dog Diseases / metabolism
  • Dog Diseases / pathology
  • Dogs
  • ErbB Receptors* / genetics
  • ErbB Receptors* / metabolism
  • Female
  • Gene Expression Regulation, Neoplastic
  • Immunohistochemistry
  • Male
  • Mutation
  • PTEN Phosphohydrolase* / genetics
  • PTEN Phosphohydrolase* / metabolism
  • Phosphatidylinositol 3-Kinases / genetics
  • Phosphatidylinositol 3-Kinases / metabolism
  • Proto-Oncogene Proteins c-akt* / genetics
  • Proto-Oncogene Proteins c-akt* / metabolism
  • Sarcoma* / genetics
  • Sarcoma* / metabolism
  • Sarcoma* / pathology
  • Sarcoma* / veterinary
  • Signal Transduction*

Substances

  • Proto-Oncogene Proteins c-akt
  • ErbB Receptors
  • PTEN Phosphohydrolase
  • Class I Phosphatidylinositol 3-Kinases
  • Phosphatidylinositol 3-Kinases