Tumor initiating activity of 5,11-dimethylchrysene and the structural requirements favoring carcinogenicity of methylated polynuclear aromatic hydrocarbons

Cancer Lett. 1979 Nov;8(1):65-70. doi: 10.1016/0304-3835(79)90024-7.

Abstract

The tumor initiating activities of 5,11-dimethylchrysene and 5-methylchrysene on mouse skin were compared. After initiating doses of 30 microgram or 10 microgram, with promotion by 3 times weekly applications of tetradecanoylphorbol acetate, both compounds were highly tumorigenic, inducing tumors in 70--85% of the treated animals. Since 5,12-dimethylchrysene had previously been shown to be only a weak tumor initiator, these results support the generalization that the structural requirements favoring carcinogenicity among the methylated chrysenes and other polynuclear aromatic hydrocarbons (PAH) are a bay region methyl group and a free peri position, both adjacent to an unsubstituted angular ring.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Chrysenes / toxicity*
  • Female
  • Methylation
  • Mice
  • Neoplasms, Experimental / chemically induced*
  • Phenanthrenes / toxicity*
  • Polycyclic Compounds / toxicity*
  • Skin Neoplasms / chemically induced
  • Structure-Activity Relationship

Substances

  • Chrysenes
  • Phenanthrenes
  • Polycyclic Compounds